Phenylalanine

Phenylalanine

SCHEMBL4614788

C[C@H](N)C(=O)O.NCC(=O)O.N[C@@H](Cc1ccccc1)C(=O)O.O=C(O)[C@@H]1CCCN1

nearest known ligand 0.49

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

SLC5A2

The experimentally established mechanism targets of Phenylalanine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC7A5 Q01650 2/20 0.49
ALPI P09923 1/20 0.49
PKM P14618 1/20 0.49
PTGS1 P23219 1/20 0.49
XIAP P98170 1/20 0.49
CTSC P53634 2/20 0.46
REN P00797 1/20 0.41
DPP4 P27487 2/20 0.39
DPP8 Q6V1X1 2/20 0.39
DPP9 Q86TI2 2/20 0.39
DPP7 Q9UHL4 2/20 0.39
ANPEP P15144 1/20 0.39
RNPEP Q9H4A4 1/20 0.39
DNPEP Q9ULA0 1/20 0.39
SLC1A3 P43003 2/20 0.39
SLC1A2 P43004 2/20 0.39
SLC1A1 P43005 2/20 0.39
SLC15A1 P46059 1/20 0.39
FAP Q12884 1/20 0.38
ACE P12821 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Phenylalanine SCHEMBL4612406 1.00 SLC7A5 (0.49) SLC7A5ALPIPKMPTGS1XIAP
Dl-Phenylalanine SCHEMBL27702676 1.00 SLC7A5 (0.49) SLC7A5ALPIPKMPTGS1XIAP
Phenylalanine SCHEMBL4405170 0.95 SLC7A5 (0.54) SLC7A5ALPIPKMPTGS1XIAP
Phenylalanine SCHEMBL3103204 0.95 SLC7A5 (0.54) SLC7A5ALPIPKMPTGS1XIAP
Dl-Phenylalanine SCHEMBL27683458 0.95 SLC7A5 (0.54) SLC7A5ALPIPKMPTGS1XIAP
Phenylalanine SCHEMBL4612447 0.95 SLC7A5 (0.54) SLC7A5ALPIPKMPTGS1XIAP
Phenylalanine SCHEMBL2764420 0.95 SLC7A5 (0.54) SLC7A5ALPIPKMPTGS1XIAP
Dl-Phenylalanine SCHEMBL29198065 0.95 SLC7A5 (0.54) SLC7A5ALPIPKMPTGS1XIAP
Dl-Phenylalanine SCHEMBL10428633 0.95 SLC7A5 (0.54) SLC7A5ALPIPKMPTGS1XIAP
Dl-Phenylalanine SCHEMBL27683462 0.95 SLC7A5 (0.54) SLC7A5ALPIPKMPTGS1XIAP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 23 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1054677-B1 COSMETIC OR DERMATOLOGICAL USE OF 7-HYDROXYLATED STEROIDS ALONE AND/OR IN COMBINATION WITH ELASTIN DERIVED PEPTIDES CONNECTIVE TISSUE IMAGINEERING (US) 2008-10-22 EP claimed
EP-1064010-A4 PEPTIDE COMPOSITIONS AND FORMULATIONS AND USE OF SAME CONNECTIVE TISSUE IMAGINEERING (US) 2004-10-06 EP claimed
US-6777389-B1 INHIBITING CUTANEOUS EFFECTS OF AGING CONNECTIVE TISSUE IMAGINEERING LLC 2004-08-17 US claimed
CN-1300220-A Peptide compositions and formulations and use of same MRS LTD (US) 2001-06-20 CN claimed
EP-1064010-A1 PEPTIDE COMPOSITIONS AND FORMULATIONS AND USE OF SAME Mrs, Llc (US) 2001-01-03 EP claimed
WO-1999045941-A1 PEPTIDE COMPOSITIONS AND FORMULATIONS AND USE OF SAME MRS, LLC (US) 1999-09-16 WO claimed
EP-1054677-B1 COSMETIC OR DERMATOLOGICAL USE OF 7-HYDROXYLATED STEROIDS ALONE AND/OR IN COMBINATION WITH ELASTIN DERIVED PEPTIDES CONNECTIVE TISSUE IMAGINEERING (US) 2008-10-22 EP disclosed
EP-1064010-B1 PEPTIDE COMPOSITIONS AND FORMULATIONS AND USE OF SAME CONNECTIVE TISSUE IMAGINEERING (US) 2008-02-20 EP disclosed
EP-1392346-A4 COMPOSITION AND METHOD FOR ENHANCING ELASTICITY OF TISSUE CONNECTIVE TISSUE IMAGINEERING (US) 2006-10-25 EP disclosed
US-6962904-B1 Elastin peptide analogs and uses thereof CONNECTIVE TISSUE IMAGINEERING (US) 2005-11-08 US disclosed
EP-1054677-A4 COSMETIC OR DERMATOLOGICAL USE OF 7-HYDROXYLATED STEROIDS ALONE AND/OR IN COMBINATION WITH ELASTIN DERIVED PEPTIDES MRS LLC (US) 2005-07-27 EP disclosed
US-20050054578-A1 Elastin peptide analogs and uses thereof SANDBERG LAWRENCE B (US) 2005-03-10 US disclosed
US-6809075-B1 Elastin peptide analogs and uses of same incombination with skin enhancing agents CONNECTIVE TISSUE IMAGINEERING LLC 2004-10-26 US disclosed
US-6506731-B1 Peptide or peptide-like compound(s) of the present invention appear to aid the elasticity and/or turgor of the skin CONNECTIVE TISSUE IMAGINEERING LLC 2003-01-14 US disclosed
WO-2001091700-A2 COMPOSITION AND METHOD FOR ENHANCING ELASTICITY OF TISSUE CONNECTIVE TISSUE IMAGINEERING LLC (US) 2001-12-06 WO disclosed
CN-1300220-A Peptide compositions and formulations and use of same MRS LTD (US) 2001-06-20 CN disclosed
EP-1064010-A1 PEPTIDE COMPOSITIONS AND FORMULATIONS AND USE OF SAME Mrs, Llc (US) 2001-01-03 EP disclosed
EP-1054677-A1 COSMETIC OR DERMATOLOGICAL USE OF 7-HYDROXYLATED STEROIDS ALONE AND/OR IN COMBINATION WITH ELASTIN DERIVED PEPTIDES Mrs, Llc (US) 2000-11-29 EP disclosed
WO-2000028996-A1 COSMETIC OR DERMATOLOGICAL USE OF 7-HYDROXYLATED STEROIDS ALONE AND/OR IN COMBINATION WITH ELASTIN DERIVED PEPTIDES MRS, LLC (US) 2000-05-25 WO disclosed
WO-1999045941-A1 PEPTIDE COMPOSITIONS AND FORMULATIONS AND USE OF SAME MRS, LLC (US) 1999-09-16 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050054578-A1 Elastin peptide analogs and uses thereof ELANE, CUTA, ENPEP SLC7A5 2652/4885ALPI 3157/4885PKM 3534/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.