SCHEMBL4618562

SCHEMBL4618562

OOC1=CCc2ccccc21

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 1/20 0.37
HPGD P15428 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
ALDH1A1 P00352 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C19 P33261 1/20 0.33
CES1 P23141 2/20 0.32
MAOA P21397 2/20 0.32
MAPT P10636 1/20 0.31
MAOB P27338 1/20 0.30
BCHE P06276 1/20 0.30
GPR84 Q9NQS5 2/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6909323 0.78 CDC25A (0.38) HTR6HPGDL3MBTL1ALDH1A1CYP1A2
SCHEMBL25176054 0.75 PTPRC (0.44) HTR6HPGDL3MBTL1ALDH1A1MAPT
SCHEMBL7633782 0.75 ALDH1A1 (0.41) HPGDALDH1A1CYP1A2MAPTMEN1
SCHEMBL7614983 0.74 HTR6 (0.34) HTR6MAOAMAOB
SCHEMBL27447443 0.72 KMT2A (0.43) HPGDALDH1A1MAPTMEN1KMT2A
SCHEMBL31072334 0.70 ALDH1A1 (0.35) HTR6L3MBTL1ALDH1A1MAPTMEN1
SCHEMBL276263 0.70 HTR6 (0.40) HTR6HPGDL3MBTL1ALDH1A1CYP1A2
SCHEMBL20219170 0.70 HTR6 (0.32) HTR6
SCHEMBL16969052 0.70 HTR6 (0.37) HTR6HPGDL3MBTL1CES1MAOA
SCHEMBL1906828 0.69 MAPT (0.33) HPGDL3MBTL1ALDH1A1CYP1A2MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1583530-A4 2-AMINOTHIAZOLE ALLOSTERIC ENHANCERS OF A1-ADENOSINE RECEPTORS UNIV VIRGINIA (US) 2008-07-23 EP disclosed
EP-1583530-A1 2-AMINOTHIAZOLE ALLOSTERIC ENHANCERS OF A1-ADENOSINE RECEPTORS UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2005-10-12 EP disclosed
WO-2003061655-A1 2-AMINOTHIAZOLE ALLOSTERIC ENHANCERS OF A1 ADENOSINE RECEPTORS UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2003-07-31 WO disclosed