SCHEMBL4618581

SCHEMBL4618581

CCOC(=O)OC1CCC2(CC1)CC(c1cccc(OC)c1)=NO2

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.43
ALDH1A1 P00352 6/20 0.42
HSD17B10 Q99714 1/20 0.42
TSHR P16473 4/20 0.41
HPGD P15428 2/20 0.41
MAPK10 P53779 1/20 0.41
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
HTT P42858 2/20 0.41
CYP3A4 P08684 3/20 0.41
CYP2C19 P33261 3/20 0.41
CYP1A2 P05177 3/20 0.41
LMNA P02545 2/20 0.41
CYP2D6 P10635 1/20 0.41
GAA P10253 1/20 0.41
KDM4E B2RXH2 1/20 0.40
GRK2 P25098 1/20 0.40
POLB P06746 1/20 0.39
APEX1 P27695 1/20 0.39
RECQL P46063 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4619940 0.87 CHRNB4 (0.41) ALDH1A1NPC1RAB9AHTTCYP2C19
SCHEMBL2208848 0.86 ALDH1A1 (0.48) NPSR1ALDH1A1HSD17B10TSHRHPGD
SCHEMBL2211286 0.81 VCP (0.45) NPSR1ALDH1A1TSHRHPGDMAPK10
SCHEMBL4351553 0.77 HTT (0.41) NPSR1ALDH1A1TSHRHPGDMAPK10
SCHEMBL15855842 0.75 NPC1 (0.51) NPSR1ALDH1A1TSHRHPGDNPC1
SCHEMBL4619812 0.75 ALDH1A1 (0.32) ALDH1A1HSD17B10GAAKDM4EPOLB
SCHEMBL2208887 0.75 CHRNB4 (0.45) ALDH1A1TSHRHPGDMAPK10NPC1
SCHEMBL5014474 0.73 TDP1 (0.47) ALDH1A1MAPK10NPC1RAB9AHTT
SCHEMBL5124433 0.73 SMN1; SMN2 (0.61) ALDH1A1HSD17B10TSHRNPC1RAB9A
SCHEMBL4620562 0.72 CHRNB4 (0.44) ALDH1A1HTTCYP2C19CYP1A2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1888542-A1 SUBSTITUTED SPIRO-COMPOUNDS AND THE USE THEREOF FOR PRODUCING MEDICAMENTS Grünenthal GmbH (DE) 2008-02-20 EP disclosed
WO-2006136245-A1 SUBSTITUTED SPIRO-COMPOUNDS AND THE USE THEREOF FOR PRODUCING MEDICAMENTS Grünenthal GmbH (DE) 2006-12-28 WO disclosed