SCHEMBL4618757

SCHEMBL4618757

[CH2]C1([CH2])COc2ccccc2C1=O

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.47
PKM P14618 1/20 0.47
CYP19A1 P11511 5/20 0.39
MAOB P27338 4/20 0.37
ALDH1A1 P00352 2/20 0.36
MEN1 O00255 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
KMT2A Q03164 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
PTGS1 P23219 1/20 0.36
PTGS2 P35354 1/20 0.36
NFKB1 P19838 1/20 0.36
NFKB2 Q00653 1/20 0.36
RELA Q04206 1/20 0.36
MAOA P21397 1/20 0.35
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9136839 0.77 PKM (0.47) TSHRPKMCYP19A1MAOBALDH1A1
SCHEMBL1133012 0.77 PKM (0.47) TSHRPKMCYP19A1MAOBALDH1A1
SCHEMBL4618755 0.77 TSHR (0.47) TSHRPKMCYP19A1MAOBALDH1A1
SCHEMBL27403505 0.77 PKM (0.47) TSHRPKMCYP19A1MAOBALDH1A1
SCHEMBL29448029 0.77 PKM (0.47) TSHRPKMCYP19A1MAOBALDH1A1
SCHEMBL4619708 0.75 CYP19A1 (0.43) CYP19A1MAOBCA1CA2CA7
SCHEMBL4620985 0.75 CYP19A1 (0.42) CYP19A1MEN1CYP2C9KMT2ACA1
SCHEMBL4619427 0.75 PARP11 (0.38) MAOBALDH1A1MEN1KMT2A
SCHEMBL29817549 0.73 TSHR (0.43) TSHRPKMCYP19A1MAOBALDH1A1
SCHEMBL3259535 0.73 NPSR1 (0.40) TSHRPKMCYP19A1MAOBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1888555-A2 SUBSTITUTED BENZO-CONDENSED CYCLOHEXANONE DERIVATIVES AND THE USE THEREOF FOR MEDICAMENT PRODUCTION Grünenthal GmbH (DE) 2008-02-20 EP claimed
WO-2006122771-A2 SUBSTITUTED BENZO-CONDENSED CYCLOHEXANONE DERIVATIVES AND THE USE THEREOF FOR MEDICAMENT PRODUCTION Grünenthal GmbH (DE) 2006-11-23 WO claimed
EP-1888555-A2 SUBSTITUTED BENZO-CONDENSED CYCLOHEXANONE DERIVATIVES AND THE USE THEREOF FOR MEDICAMENT PRODUCTION Grünenthal GmbH (DE) 2008-02-20 EP disclosed
WO-2006122771-A2 SUBSTITUTED BENZO-CONDENSED CYCLOHEXANONE DERIVATIVES AND THE USE THEREOF FOR MEDICAMENT PRODUCTION Grünenthal GmbH (DE) 2006-11-23 WO disclosed