SCHEMBL461891

SCHEMBL461891

Fc1cc(Cl)ccc1CC(F)(F)F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 3/20 0.40
TP53 P04637 1/20 0.40
HTR1A P08908 1/20 0.40
HTR7 P34969 1/20 0.40
HTR6 P50406 1/20 0.40
NR1H2 P55055 1/20 0.38
NR1H3 Q13133 1/20 0.38
CXCR3 P49682 3/20 0.38
IDO1 P14902 2/20 0.38
GGPS1 O95749 1/20 0.37
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
MAPK1 P28482 1/20 0.36
CYP2C19 P33261 1/20 0.36
SLC6A4 P31645 3/20 0.36
KCNH2 Q12809 2/20 0.36
GRM2 Q14416 1/20 0.36
VNN1 O95497 1/20 0.36
ERCC1 P07992 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20256821 0.85 MPO (0.40) HTR2AIDO1GGPS1CYP1A2CYP3A4
SCHEMBL9917350 0.82 HTR2A (0.39) HTR2ATP53HTR1AHTR7HTR6
SCHEMBL3799579 0.79 HTR2A (0.50) HTR2ATP53HTR1AHTR7HTR6
SCHEMBL30090066 0.79 NR3C1 (0.38) HTR2ATP53HTR1AHTR7HTR6
SCHEMBL19030566 0.79 NR3C1 (0.38) HTR2ATP53HTR1AHTR7HTR6
SCHEMBL1381639 0.78 IDO1 (0.50) HTR2AIDO1ALDH1A1HTR2C
SCHEMBL19030189 0.78 NR3C1 (0.41) HTR2ATP53HTR1AHTR7HTR6
SCHEMBL4604208 0.78 KMT2A (0.48) HTR2ATP53HTR1AHTR7HTR6
SCHEMBL5717224 0.77 GRM2 (0.38) HTR2ATP53HTR1AHTR7HTR6
SCHEMBL12841965 0.77 HTR2A (0.36) HTR2ATP53HTR1AHTR7HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022228490-A1 POLYCYCLIC DERIVATIVE MODULATOR, AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海翰森生物医药科技有限公司 2022-11-03 WO disclosed
EP-2595984-A1 MICROBICIDES Syngenta Participations AG (CH) 2013-05-29 EP disclosed
EP-2595985-A1 ISOXAZOLE, ISOTHIAZOLE, FURANE AND THIOPHENE COMPOUNDS AS MICROBICIDES Syngenta Participations AG (CH) 2013-05-29 EP disclosed
WO-2012010568-A1 MICROBICIDES SYNGENTA PARTICIPATIONS AG (CH) 2012-01-26 WO disclosed
WO-2012010567-A1 ISOXAZOLE, ISOTHIAZOLE, FURANE AND THIOPHENE COMPOUNDS AS MICROBICIDES SYNGENTA PARTICIPATIONS AG (CH) 2012-01-26 WO disclosed