SCHEMBL4619458

SCHEMBL4619458

NS(=O)(=O)c1ccc(-c2cc(-c3ccc(F)c(C(F)(F)F)c3)on2)cc1.NS(=O)(=O)c1ccc(-c2cc(-c3ccc(OCC(F)(F)F)c(C(F)(F)F)c3)on2)cc1

nearest known ligand 0.55

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 6/20 0.55
S1PR1 P21453 5/20 0.54
KIF11 P52732 1/20 0.42
PTGS1 P23219 4/20 0.38
AAK1 Q2M2I8 5/20 0.37
CYP3A4 P08684 1/20 0.36
LMNA P02545 1/20 0.36
TP53 P04637 1/20 0.36
THRB P10828 1/20 0.36
MPL P40238 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4931412 0.95 S1PR1 (0.58) PTGS2S1PR1KIF11PTGS1AAK1
SCHEMBL4618798 0.90 PTGS2 (0.67) PTGS2S1PR1KIF11PTGS1LMNA
SCHEMBL4618115 0.72 S1PR1 (0.67) S1PR1KIF11
SCHEMBL20615395 0.70 S1PR1 (1.00) S1PR1
SCHEMBL3275084 0.67 S1PR1 (0.59) S1PR1
SCHEMBL6733221 0.67 PTGS2 (0.65) PTGS2KIF11PTGS1
SCHEMBL22981523 0.67 SGK1 (0.43) PTGS2S1PR1KIF11MPL
SCHEMBL6728375 0.66 KIF11 (0.58) PTGS2KIF11PTGS1
SCHEMBL6728905 0.66 PTGS2 (0.66) PTGS2KIF11PTGS1
SCHEMBL29793217 0.66 KIF11 (0.60) PTGS2KIF11PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1893591-A1 POLYCYCLIC OXADIAZOLES OR I SOXAZOLES AND THEIR USE AS SlP RECEPTOR LIGANDS Novartis AG (CH) 2008-03-05 EP disclosed
WO-2006131336-A1 POLYCYCLIC OXADIAZOLES OR I SOXAZOLES AND THEIR USE AS SlP RECEPTOR LIGANDS NOVARTIS AG (CH) 2006-12-14 WO disclosed