SCHEMBL4620344

SCHEMBL4620344

CCCCC1(CCCC)NSC2=C(C(=O)[C@@H](SC)C(OCC(=O)N[C@@H](C(=O)NCCCC(=O)O)c3ccccc3)=C2)N(c2ccccc2)C1=O

nearest known ligand 0.34

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CTSD P07339 3/20 0.34
NR1H4 Q96RI1 1/20 0.32
LTA4H P09960 1/20 0.30
ALDH1A1 P00352 1/20 0.30
PTPN1 P18031 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3836011 0.97 NR1H4 (0.34) CTSDNR1H4
SCHEMBL4664295 0.96 NR1H4 (0.37) CTSDNR1H4
SCHEMBL4596808 0.94 NR1H4 (0.36) CTSDNR1H4
SCHEMBL3834127 0.93 NR1H4 (0.38) CTSDNR1H4
SCHEMBL14895745 0.93 NR1H4 (0.33) CTSDNR1H4
SCHEMBL5709136 0.92 NR1H4 (0.35) CTSDNR1H4
SCHEMBL6157024 0.90 NR1H4 (0.34) CTSDNR1H4
SCHEMBL5709156 0.89 CTSD (0.33) CTSDNR1H4
SCHEMBL4617149 0.89 NR1H4 (0.35) CTSDNR1H4
SCHEMBL14895557 0.89 NR1H4 (0.42) CTSDNR1H4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1885694-A2 4-BIARYLYL-1-PHENYLAZETIDIN-2-ONES Microbia, Inc. (US) 2008-02-13 EP disclosed
EP-1851197-A2 PHENYLAZETIDINONE DERIVATIVES Microbia, Inc. (US) 2007-11-07 EP disclosed
WO-2006124713-A2 4-BIARYLYL-1-PHENYLAZETIDIN-2-ONES MICROBIA, INC. (US) 2006-11-23 WO disclosed
WO-2006086562-A2 PHENYLAZETIDINONE DERIVATIVES MICROBIA, INC. (US) 2006-08-17 WO disclosed
EP-1572626-A1 THERAPEUTIC AGENTS Astrazeneca AB (SE) 2005-09-14 EP disclosed
WO-2004056748-A1 THERAPEUTIC AGENTS ASTRAZENECA AB (SE) 2004-07-08 WO disclosed