SCHEMBL4620423

SCHEMBL4620423

[CH]C1([CH])COc2c(C)cc(Cc3ccccc3)cc2C1=O

nearest known ligand 0.35

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 4/20 0.35
NQO1 P15559 1/20 0.32
EDNRA P25101 2/20 0.31
EDNRB P24530 1/20 0.31
PARP11 Q9NR21 1/20 0.31
PTPN2 P17706 2/20 0.31
PTPN6 P29350 2/20 0.31
CALM1 P0DP23 1/20 0.31
HMGB1 P09429 1/20 0.31
CXCL12 P48061 1/20 0.31
CNR2 P34972 2/20 0.30
GPR55 Q9Y2T6 2/20 0.30
IDH1 O75874 3/20 0.30
MAOB P27338 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4620426 0.85 PTPN1 (0.35) PTPN1NQO1PARP11PTPN2PTPN6
SCHEMBL2156032 0.79 PTPN1 (0.38) PTPN1NQO1PTPN2PTPN6HMGB1
SCHEMBL4619425 0.77 PARP11 (0.38) EDNRAEDNRBPARP11CALM1IDH1
SCHEMBL2156037 0.77 PRKCA (0.36) PTPN1EDNRAEDNRBIDH1
SCHEMBL2435285 0.64 PTPN1 (0.37) PTPN1NQO1PTPN2PTPN6CALM1
SCHEMBL8100218 0.61 CALM1 (0.55) NQO1CALM1HMGB1CXCL12IDH1
SCHEMBL28888543 0.60 CALM1 (0.52) PTPN1PTPN2PTPN6CALM1HMGB1
SCHEMBL27509240 0.60 CALM1 (0.52) CALM1IDH1
SCHEMBL9480008 0.60 HMGB1 (0.55) PTPN1NQO1PTPN2PTPN6CALM1
SCHEMBL10525358 0.59 PARP11 (0.44) PTPN1PARP11CALM1IDH1MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1888555-A2 SUBSTITUTED BENZO-CONDENSED CYCLOHEXANONE DERIVATIVES AND THE USE THEREOF FOR MEDICAMENT PRODUCTION Grünenthal GmbH (DE) 2008-02-20 EP claimed
WO-2006122771-A2 SUBSTITUTED BENZO-CONDENSED CYCLOHEXANONE DERIVATIVES AND THE USE THEREOF FOR MEDICAMENT PRODUCTION Grünenthal GmbH (DE) 2006-11-23 WO claimed
EP-1888555-A2 SUBSTITUTED BENZO-CONDENSED CYCLOHEXANONE DERIVATIVES AND THE USE THEREOF FOR MEDICAMENT PRODUCTION Grünenthal GmbH (DE) 2008-02-20 EP disclosed
WO-2006122771-A2 SUBSTITUTED BENZO-CONDENSED CYCLOHEXANONE DERIVATIVES AND THE USE THEREOF FOR MEDICAMENT PRODUCTION Grünenthal GmbH (DE) 2006-11-23 WO disclosed