SCHEMBL4620526

SCHEMBL4620526

CN(C)C(=O)c1ccc([N+](=O)[O-])cc1S(N)(=O)=O

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.62
ALDH1A1 P00352 5/20 0.48
CYP3A4 P08684 2/20 0.48
ALOX15 P16050 2/20 0.48
PDE2A O00408 1/20 0.48
PDE5A O76074 1/20 0.48
NFKB1 P19838 1/20 0.48
APEX1 P27695 1/20 0.48
PDE4A P27815 1/20 0.48
BLM P54132 1/20 0.48
PDE1B Q01064 1/20 0.48
PMP22 Q01453 1/20 0.48
PDE4B Q07343 1/20 0.48
PDE4D Q08499 1/20 0.48
PDE7A Q13946 1/20 0.48
PDE1C Q14123 1/20 0.48
PDE7B Q9NP56 1/20 0.48
KMT2A Q03164 3/20 0.46
HPGD P15428 2/20 0.46
MEN1 O00255 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Potassium Ion SCHEMBL2975282 0.87 L3MBTL1 (0.60) L3MBTL1ALDH1A1CYP3A4ALOX15PDE2A
SCHEMBL2980353 0.87 L3MBTL1 (0.60) L3MBTL1ALDH1A1CYP3A4ALOX15PDE2A
Potassium Ion SCHEMBL2975285 0.87 L3MBTL1 (0.60) L3MBTL1ALDH1A1CYP3A4ALOX15PDE2A
SCHEMBL2970340 0.86 L3MBTL1 (0.58) L3MBTL1ALDH1A1CYP3A4ALOX15PDE2A
SCHEMBL2970344 0.86 L3MBTL1 (0.58) L3MBTL1ALDH1A1CYP3A4ALOX15PDE2A
Potassium SCHEMBL2975289 0.86 L3MBTL1 (0.58) L3MBTL1ALDH1A1CYP3A4ALOX15PDE2A
SCHEMBL6105510 0.86 L3MBTL1 (0.58) L3MBTL1ALDH1A1CYP3A4ALOX15PDE2A
SCHEMBL2970353 0.86 L3MBTL1 (0.58) L3MBTL1ALDH1A1CYP3A4ALOX15PDE2A
SCHEMBL8536343 0.82 ALDH1A1 (0.61) ALDH1A1CYP3A4ALOX15KMT2AMEN1
SCHEMBL7685851 0.81 L3MBTL1 (0.53) L3MBTL1ALDH1A1CYP3A4ALOX15PDE2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 35 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112125828-B Synthetic method of foramsulfuron intermediate 江苏省农用激素工程技术研究中心有限公司 2022-05-06 CN claimed
CN-110437112-B Preparation method of formamidosulfuron or derivative intermediate thereof 河北兴柏农业科技有限公司 2021-08-17 CN claimed
CN-112125828-A Synthetic method of foramsulfuron intermediate 江苏省农用激素工程技术研究中心有限公司 2020-12-25 CN claimed
CN-110437112-A A kind of preparation method of formamido group Sulfometuron Methyl or derivatives thereof intermediate HEBEI XINGBAI AGRICULTURAL TECH CO LTD 2019-11-12 CN claimed
CN-116903545-A Synthesis method of formamide sulfosulfuron 江苏省农用激素工程技术研究中心有限公司 2023-10-20 CN disclosed
CN-112125828-B Synthetic method of foramsulfuron intermediate 江苏省农用激素工程技术研究中心有限公司 2022-05-06 CN disclosed
CN-112125828-B Synthetic method of foramsulfuron intermediate 江苏省农用激素工程技术研究中心有限公司 2022-05-06 CN disclosed
CN-113735782-A Preparation method of foramsulfuron 安徽丰乐农化有限责任公司 2021-12-03 CN disclosed
CN-110437112-B Preparation method of formamidosulfuron or derivative intermediate thereof 河北兴柏农业科技有限公司 2021-08-17 CN disclosed
CN-110437112-B Preparation method of formamidosulfuron or derivative intermediate thereof 河北兴柏农业科技有限公司 2021-08-17 CN disclosed
CN-112125828-A Synthetic method of foramsulfuron intermediate 江苏省农用激素工程技术研究中心有限公司 2020-12-25 CN disclosed
CN-112125828-A Synthetic method of foramsulfuron intermediate 江苏省农用激素工程技术研究中心有限公司 2020-12-25 CN disclosed
US-6365739-B1 REACTION OF AMINOPYRAMIDINE WITH PHOSGENE TO FORM ISOCYANATO PYRIMIDINE HOECHST SCHERING AGREVO GMBH (DE) 2002-04-02 US disclosed
EP-0858447-B1 METHODS OF PRODUCING AMINOPHENYLSULPHONYL CARBAMIDES AND INTERMEDIATE PRODUCTS FOR USE IN THE PROCESS AVENTIS CROPSCIENCE GMBH (DE) 2002-01-09 EP disclosed
CN-1311782-A Method for producing 4,6-disubstituted 2-isocyanatopyrimidines and to their use as intermediate products for active ingredient syntheses AVENTIES CROPS SCIENCE GMBH (DE) 2001-09-05 CN disclosed
EP-1097144-A1 METHOD FOR PRODUCING 4,6-DISUBSTITUTED 2-ISOCYANATOPYRIMIDINES AND TO THEIR USE AS INTERMEDIATE PRODUCTS FOR ACTIVE INGREDIENT SYNTHESES Aventis CropScience GmbH (DE) 2001-05-09 EP disclosed
WO-2000005220-A1 METHOD FOR PRODUCING 4,6-DISUBSTITUTED 2-ISOCYANATOPYRIMIDINES AND TO THEIR USE AS INTERMEDIATE PRODUCTS FOR ACTIVE INGREDIENT SYNTHESES AVENTIS CROPSCIENCE GMBH (DE) 2000-02-03 WO disclosed
CN-1202884-A Process for preparing aminophenylsulfonylureas, and intermediates for their preparation HOECHST SCHERING AGREVO GMBH (DE) 1998-12-23 CN disclosed
EP-0858447-A1 METHODS OF PRODUCING AMINOPHENYLSULPHONYL CARBAMIDES AND INTERMEDIATE PRODUCTS FOR USE IN THE PROCESS Hoechst Schering AgrEvo GmbH (DE) 1998-08-19 EP disclosed
WO-1997016419-A1 METHODS OF PRODUCING AMINOPHENYLSULPHONYL CARBAMIDES AND INTERMEDIATE PRODUCTS FOR USE IN THE PROCESS HOECHST SCHERING AGREVO GMBH (DE) 1997-05-09 WO disclosed