SCHEMBL4620748

SCHEMBL4620748

O=C(Cn1c(=O)oc2ccccc21)N[C@@H](CCCSCC(=O)C(F)(F)F)C(=O)NCC(O)c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.40
CYP1A2 P05177 3/20 0.40
CYP2C19 P33261 3/20 0.40
POLB P06746 3/20 0.40
CYP3A4 P08684 2/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2D6 P10635 2/20 0.39
PKM P14618 1/20 0.39
KMT2A Q03164 3/20 0.38
IDO1 P14902 2/20 0.38
CDYL2 Q8N8U2 3/20 0.38
CDYL Q9Y232 3/20 0.38
CDY1; CDY1B Q9Y6F8 3/20 0.38
CBX7 O95931 2/20 0.38
RECQL P46063 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
ALDH1A1 P00352 1/20 0.38
MEN1 O00255 1/20 0.38
TP53 P04637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4621007 0.83 POLB (0.51) LMNACYP1A2CYP2C19POLBCYP3A4
Trifluoroacetic Acid SCHEMBL4618886 0.80 POLB (0.38) LMNACYP1A2CYP2C19POLBCYP3A4
SCHEMBL4158065 0.80 CES1 (0.45) KMT2AALDH1A1
SCHEMBL4161122 0.78 NPC1 (0.46) KMT2ASMN1; SMN2MEN1
Trifluoroacetic Acid SCHEMBL4622701 0.78 CHRM1 (0.46)
Trifluoroacetic Acid SCHEMBL4158022 0.77 HDAC1 (0.38) SMN1; SMN2
SCHEMBL4171678 0.76 HPGD (0.40) CYP1A2CYP2C19CYP3A4KMT2AIDO1
SCHEMBL4151885 0.73 KMT2A (0.43) LMNACYP1A2CYP2C19POLBCYP3A4
SCHEMBL4159834 0.73 EPHX2 (0.43) LMNACYP1A2CYP2C19CYP3A4CYP2C9
Trifluoroacetic Acid SCHEMBL4171443 0.72 CHRM1 (0.38) LMNACYP1A2CYP2C19POLBCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1945609-A2 AMINO ACID DERIVATIVES AS HISTONE DEACETYLASE (HDAC) INHIBITORS ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI S.P.A. (IT) 2008-07-23 EP disclosed
WO-2007029036-A2 AMINO ACID DERIVATIVES AS HISTONE DEACETYLASE (HDAC) INHIBITORS ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI SPA (IT) 2007-03-15 WO disclosed