SCHEMBL4621840

SCHEMBL4621840

CC(C)(Cc1ccccc1)N(C(=O)c1ccc(Br)cc1)[C@@H](CCC(N)=O)C(=O)O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.37
HSP90AA1 P07900 1/20 0.37
MEN1 O00255 3/20 0.37
MAPK1 P28482 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
TDP1 Q9NUW8 1/20 0.35
ITK Q08881 1/20 0.35
CHRM2 P08172 1/20 0.33
CHRM3 P20309 1/20 0.33
MLYCD O95822 2/20 0.33
TMEM97 Q5BJF2 1/20 0.33
SIGMAR1 Q99720 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
ALOX15 P16050 1/20 0.33
TSHR P16473 1/20 0.33
CYP2C19 P33261 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2245867 0.90 MMP2 (0.40) SMN1; SMN2L3MBTL1ITKALDH1A1
SCHEMBL2245162 0.87 ERN1 (0.36) KMT2AMEN1ALDH1A1LMNAKIF11
SCHEMBL2244927 0.87 PPARG (0.37) L3MBTL1TDP1ALDH1A1LMNATSHR
SCHEMBL2245097 0.87 KMT2A (0.37) KMT2AHSP90AA1MEN1MAPK1SMN1; SMN2
SCHEMBL2247320 0.86 MMP2 (0.35) KMT2AMEN1ALDH1A1LMNACYP3A4
SCHEMBL2245193 0.86 MMP2 (0.43) KMT2AMEN1MAPK1TDP1ALDH1A1
SCHEMBL2245812 0.85 HDAC1 (0.37) SMN1; SMN2L3MBTL1ALDH1A1
SCHEMBL27708299 0.85 RORC (0.35) ITKCYP3A4
SCHEMBL2247635 0.84 MCHR1 (0.36) ALDH1A1CYP3A4ALOX15
SCHEMBL2252602 0.83 TP53 (0.35) L3MBTL1ALDH1A1LMNAKIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101223130-A Glutamate aggrecanase inhibitors WYETH CORP (US) 2008-07-16 CN claimed
CN-101223130-A Glutamate aggrecanase inhibitors WYETH CORP (US) 2008-07-16 CN disclosed
EP-1902014-A2 GLUTAMATE AGGRECANASE INHIBITORS Wyeth (US) 2008-03-26 EP disclosed
WO-2007008994-A2 GLUTAMATE AGGRECANASE INHIBITORS WYETH (US) 2007-01-18 WO disclosed