SCHEMBL4623218

SCHEMBL4623218

CC1NC(=O)Nc2ccc(-c3ccc(C(F)(F)F)cc3)cc21.O=C1Nc2ccc(-c3ccc(C(F)(F)F)cc3)cc2CO1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 2/20 0.47
CYP11B1 P15538 3/20 0.46
CYP11B2 P19099 3/20 0.46
TDP2 O95551 1/20 0.39
CHRNB2 P17787 1/20 0.34
CHRNA4 P43681 1/20 0.34
SYK P43405 2/20 0.34
CTSC P53634 1/20 0.34
PDE3B Q13370 3/20 0.33
PDE3A Q14432 3/20 0.33
BRD4 O60885 1/20 0.32
BRD2 P25440 1/20 0.32
BRD3 Q15059 1/20 0.32
SIGMAR1 Q99720 1/20 0.32
PARP1 P09874 1/20 0.31
PARP2 Q9UGN5 1/20 0.31
GRIA1 P42261 1/20 0.31
CDK2 P24941 2/20 0.31
AKT1 P31749 2/20 0.31
CDK1 P06493 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4595017 0.91 CYP11B1 (0.41) KIF11CYP11B1CYP11B2TDP2SYK
SCHEMBL4898275 0.86 KIF11 (0.48) KIF11TDP2CHRNB2CHRNA4PDE3B
SCHEMBL4596312 0.84 KIF11 (0.63) KIF11CYP11B1CYP11B2TDP2CHRNB2
SCHEMBL4596036 0.71 KIF11 (0.45) KIF11TDP2CHRNB2CHRNA4BRD4
SCHEMBL19187758 0.71 CYP11B1 (0.60) KIF11CYP11B1CYP11B2SYKCTSC
SCHEMBL4596871 0.69 KIF11 (0.59) KIF11CYP11B1CYP11B2TDP2CHRNB2
SCHEMBL4596644 0.69 KIF11 (0.70) KIF11CYP11B1CYP11B2TDP2PDE3B
SCHEMBL4596437 0.69 KIF11 (0.65) KIF11CYP11B1CYP11B2TDP2CHRNB2
SCHEMBL1903306 0.67 KIF11 (0.80) KIF11CYP11B1CYP11B2TDP2PDE3B
SCHEMBL2054589 0.67 CYP11B1 (0.48) KIF11CYP11B1CYP11B2SYKPDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874753-A2 COMPOUNDS, COMPOSITIONS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2008-01-09 EP disclosed
WO-2006113432-A2 COMPOUNDS, COMPOSITIONS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2006-10-26 WO disclosed