SCHEMBL4626229

SCHEMBL4626229

Cc1cc(C)c(-c2cn(C)c3nc[nH]c(=O)c23)c(C)c1

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CRHR1 P34998 5/20 0.47
MAPT P10636 5/20 0.44
LMNA P02545 3/20 0.44
KMT2A Q03164 1/20 0.44
HTT P42858 2/20 0.44
PARP1 P09874 2/20 0.43
BRD4 O60885 2/20 0.42
SRC P12931 1/20 0.40
ALDH1A1 P00352 1/20 0.37
PKM P14618 1/20 0.37
GAA P10253 1/20 0.36
BCAT2 O15382 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2072133 0.78 CRHR1 (0.51) CRHR1
SCHEMBL15265113 0.75 SRC (0.68) MAPTLMNAKMT2AHTTBRD4
SCHEMBL2070607 0.71 CRHR1 (0.65) CRHR1
SCHEMBL20224829 0.71 PARP1 (0.44) MAPTLMNAKMT2AHTTPARP1
SCHEMBL15265574 0.71 ALDH1A1 (0.44) MAPTLMNAKMT2AHTTPARP1
SCHEMBL20224898 0.71 CDK2 (0.44) MAPTLMNAKMT2AHTTPARP1
SCHEMBL2069734 0.70 CRHR1 (0.65) CRHR1
SCHEMBL13838861 0.70 CRHR1 (0.51) CRHR1ALDH1A1GAA
SCHEMBL2070441 0.68 CRHR1 (0.54) CRHR1
SCHEMBL2071976 0.68 CRHR1 (0.60) CRHR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1732541-A4 CYCLIC COMPOUNDS TAKEDA PHARMACEUTICAL (JP) 2008-03-05 EP disclosed
EP-1732541-A2 CYCLIC COMPOUNDS Takeda Pharmaceutical Company Limited (JP) 2006-12-20 EP disclosed
WO-2005099688-A2 CYCLIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2005-10-27 WO disclosed