SCHEMBL4627344

SCHEMBL4627344

Clc1cccc(Cl)c1-c1ccc2cccc(OCc3ccccc3)c2n1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.48
MAPT P10636 2/20 0.48
CCR6 P51684 1/20 0.48
MEN1 O00255 5/20 0.48
KMT2A Q03164 5/20 0.48
PIM1 P11309 2/20 0.47
PIM2 Q9P1W9 2/20 0.47
HPGD P15428 4/20 0.47
ALDH1A1 P00352 2/20 0.47
HTT P42858 1/20 0.47
BDKRB2 P30411 1/20 0.45
NPC1 O15118 3/20 0.45
RAB9A P51151 3/20 0.45
HTR1A P08908 1/20 0.44
ADRA1D P25100 1/20 0.44
ADRA1A P35348 1/20 0.44
ADRA1B P35368 1/20 0.44
HDAC3 O15379 2/20 0.43
HDAC4 P56524 2/20 0.43
HDAC1 Q13547 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL729315 0.81 MEN1 (0.54) KDM4EMAPTCCR6MEN1KMT2A
SCHEMBL4626663 0.79 HTR1A (0.51) KDM4EMAPTCCR6MEN1KMT2A
SCHEMBL9951781 0.77 MEN1 (0.55) KDM4EMAPTCCR6MEN1KMT2A
SCHEMBL28622872 0.76 MEN1 (0.51) KDM4EMAPTCCR6MEN1KMT2A
SCHEMBL3949886 0.76 MEN1 (0.78) KDM4EMAPTCCR6MEN1KMT2A
SCHEMBL18438857 0.76 MEN1 (0.61) KDM4EMAPTCCR6MEN1KMT2A
SCHEMBL28284853 0.76 MEN1 (0.59) KDM4EMAPTCCR6MEN1KMT2A
SCHEMBL1012890 0.76 NCF1 (0.63) KDM4EMAPTCCR6
SCHEMBL731221 0.76 KDM4E (0.56) KDM4EMAPTCCR6MEN1KMT2A
SCHEMBL19830909 0.75 MEN1 (0.53) KDM4EMAPTCCR6MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501801-B1 2,6-QUINOLINYL AND 2,6-NAPHTHYL DERIVATIVES AND THEIR USE IN THE TREATMENT OF VLA-4 DEPENDENT DISEASES UCB PHARMA SA (BE) 2008-01-23 EP claimed