SCHEMBL4627746

SCHEMBL4627746

CCCC(CCC(=O)Br)c1cccc2c1CC(C(=O)OCC)=CN2

nearest known ligand 0.32

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.32
CA12 O43570 1/20 0.31
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
CA7 P43166 1/20 0.31
CA9 Q16790 1/20 0.31
CA14 Q9ULX7 1/20 0.31
POLB P06746 1/20 0.31
CYP1A2 P05177 1/20 0.30
KDM4E B2RXH2 2/20 0.30
MEN1 O00255 1/20 0.30
NPC1 O15118 1/20 0.30
ALDH1A1 P00352 1/20 0.30
LMNA P02545 1/20 0.30
GLA P06280 1/20 0.30
GAA P10253 1/20 0.30
MAPT P10636 1/20 0.30
HPGD P15428 1/20 0.30
RAB9A P51151 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4626316 0.78 KDM4E (0.32) KDM4EMEN1NPC1ALDH1A1LMNA
SCHEMBL29008018 0.69 TSHR (0.45) CA12CA1CA2CA7CA9
Hydrochloric Acid SCHEMBL29008069 0.68 TSHR (0.44) CA12CA1CA2CA7CA9
SCHEMBL9797391 0.60 KDM4E (0.48) CA12CA1CA2CA7CA9
SCHEMBL7425087 0.60 KDM4E (0.59) CA12CA1CA2CA7CA9
SCHEMBL29105832 0.60 TSHR (0.59) CA2POLBKDM4EALDH1A1LMNA
SCHEMBL30585963 0.59 BRD4 (0.42) CA12CA1CA2CA7CA9
SCHEMBL9748650 0.58 KMT2A (0.40) CA12CA1CA2CA7CA9
SCHEMBL30958562 0.58 KDM4E (0.47) POLBKDM4EMEN1ALDH1A1LMNA
SCHEMBL6026672 0.58 ATM (0.41) KDM4EMEN1NPC1ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1732541-A4 CYCLIC COMPOUNDS TAKEDA PHARMACEUTICAL (JP) 2008-03-05 EP disclosed
EP-1732541-A2 CYCLIC COMPOUNDS Takeda Pharmaceutical Company Limited (JP) 2006-12-20 EP disclosed
WO-2005099688-A2 CYCLIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2005-10-27 WO disclosed