SCHEMBL4628522

SCHEMBL4628522

CC(Br)C(=O)Cl.CC(Br)C(=O)Nc1cccc(Br)c1O

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CXCR2 P25025 10/20 0.43
CXCR1 P25024 9/20 0.43
L3MBTL1 Q9Y468 2/20 0.40
ATM Q13315 1/20 0.40
TP53 P04637 2/20 0.39
GAA P10253 1/20 0.39
ANPEP P15144 1/20 0.38
MDM4 O15151 1/20 0.37
HTT P42858 2/20 0.36
MEN1 O00255 1/20 0.36
NPC1 O15118 1/20 0.36
LMNA P02545 1/20 0.36
RAB9A P51151 1/20 0.36
KMT2A Q03164 1/20 0.36
CETP P11597 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2070180 0.94 ATM (0.43) CXCR2CXCR1L3MBTL1ATMTP53
SCHEMBL4971514 0.82 HTT (0.44) CXCR2CXCR1L3MBTL1ATMTP53
SCHEMBL23705971 0.74 RXFP1 (0.51) CXCR2CXCR1GAAMEN1NPC1
SCHEMBL4969475 0.73 CXCR2 (0.46) CXCR2CXCR1L3MBTL1ATMGAA
SCHEMBL14157620 0.72 LMNA (0.46) CXCR2CXCR1L3MBTL1HTTMEN1
SCHEMBL4675699 0.70 PDK1 (0.50) CXCR2CXCR1HTTMEN1NPC1
SCHEMBL30797039 0.70 PDK1 (0.50) CXCR2CXCR1HTTMEN1NPC1
SCHEMBL11731600 0.69 NPC1 (0.60) GAAANPEPHTTNPC1LMNA
SCHEMBL4969948 0.69 CXCR2 (0.45) CXCR2CXCR1TP53MDM4HTT
SCHEMBL3742208 0.68 SMN1; SMN2 (0.63) GAAHTTMEN1NPC1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1732541-A4 CYCLIC COMPOUNDS TAKEDA PHARMACEUTICAL (JP) 2008-03-05 EP disclosed
EP-1732541-A2 CYCLIC COMPOUNDS Takeda Pharmaceutical Company Limited (JP) 2006-12-20 EP disclosed
WO-2005099688-A2 CYCLIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2005-10-27 WO disclosed