SCHEMBL4628997

SCHEMBL4628997

CCCCCC([Si](C)(C)Cl)[Si](C)(C)Cl

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 1/20 0.40
FDPS P14324 4/20 0.39
LMNA P02545 1/20 0.37
DNM1 Q05193 2/20 0.36
TSHR P16473 2/20 0.35
THRB P10828 1/20 0.35
GPR84 Q9NQS5 3/20 0.33
ALDH1A1 P00352 1/20 0.33
SPHK1 Q9NYA1 1/20 0.33
FFAR1 O14842 1/20 0.33
CA1 P00915 1/20 0.33
MAPT P10636 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2381454 0.97 FDPS (0.41) OPRM1FDPSLMNADNM1TSHR
SCHEMBL4262636 0.84 OPRM1 (0.40) OPRM1FDPSLMNADNM1TSHR
SCHEMBL671491 0.83 OPRM1 (0.43) OPRM1FDPSLMNADNM1TSHR
SCHEMBL1031063 0.82 FDPS (0.41) OPRM1FDPSLMNADNM1TSHR
SCHEMBL14995732 0.81 FDPS (0.44) OPRM1FDPSLMNADNM1TSHR
SCHEMBL6512567 0.81 FDPS (0.44) OPRM1FDPSLMNADNM1TSHR
SCHEMBL337206 0.81 FDPS (0.44) OPRM1FDPSLMNADNM1TSHR
SCHEMBL11347774 0.81 FDPS (0.44) OPRM1FDPSLMNADNM1TSHR
SCHEMBL785693 0.81 FDPS (0.44) OPRM1FDPSLMNADNM1TSHR
SCHEMBL5163533 0.78 OPRM1 (0.43) OPRM1FDPSLMNADNM1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013079939-A2 OSCILLATOR SPRING COMPOSITION AND METHOD FOR FABRICATING AN OSCILLATOR SPRING CARBONTIME LIMITED (GB) 2013-06-06 WO claimed
EP-1919926-A2 PROCESSES FOR THE PRODUCTION OF POLYCYCLIC FUSED RING COMPOUNDS Florida State University Research Foundation, Inc. (US) 2008-05-14 EP claimed
EP-1893594-A2 PROCESSES FOR THE PREPARATION OF PACLITAXEL Florida State University Research Foundation, Inc. (US) 2008-03-05 EP claimed
EP-1891033-A2 PROCESSES FOR THE PREPARATION OF DOCETAXEL Florida State University Research Foundation, Inc. (US) 2008-02-27 EP claimed
WO-2006135692-A2 PROCESSES FOR THE PREPARATION OF DOCETAXEL FLORIDA STATE UNIVERSITY RESEARCH FOUNDATION, INC. (US) 2006-12-21 WO claimed
WO-2006135656-A2 PROCESSES FOR THE PREPARATION OF PACLITAXEL FLORIDA STATE UNIVERSITY RESEARCH FOUNDATION, INC. (US) 2006-12-21 WO claimed
WO-2006135655-A2 PROCESSES FOR THE PRODUCTION OF POLYCYCLIC FUSED RING COMPOUNDS FLORIDA STATE UNIVERSITY RESEARCH FOUNDATION, INC. (US) 2006-12-21 WO claimed
EP-2785695-A1 NEW BICYCLIC DIHYDROISOQUINOLINE-1-ONE DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 2014-10-08 EP disclosed
WO-2013079452-A1 NEW BICYCLIC DIHYDROISOQUINOLINE-1-ONE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2013-06-06 WO disclosed
WO-2013079939-A2 OSCILLATOR SPRING COMPOSITION AND METHOD FOR FABRICATING AN OSCILLATOR SPRING CARBONTIME LIMITED (GB) 2013-06-06 WO disclosed
EP-1543054-A1 POLYMERS WITH SOFT SEGMENTS CONTAINING SILANE-CONTAINING GROUPS, MEDICAL DEVICES, AND METHODS Medtronic, Inc. (US) 2005-06-22 EP disclosed
WO-2004026933-A1 POLYMERS WITH SOFT SEGMENTS CONTAINING SILANE-CONTAINING GROUPS, MEDICAL DEVICES, AND METHODS MEDTRONIC, INC. (US) 2004-04-01 WO disclosed
WO-2003035252-A1 CHEMICAL MODIFICATION OF PARTICLE SURFACES BY CROSS-LINKING MERCK PATENT GMBH (DE) 2003-05-01 WO disclosed