SCHEMBL4629623

SCHEMBL4629623

O=[C]C1CCN(NC(=O)c2ccccc2)C1

nearest known ligand 0.54

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.54
CTSL P07711 4/20 0.44
CTSB P07858 4/20 0.44
CTSK P43235 4/20 0.44
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
CYP2C9 P11712 2/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C19 P33261 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.39
LMNA P02545 1/20 0.38
MAPK1 P28482 1/20 0.38
GAA P10253 1/20 0.38
MAPT P10636 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28138491 0.75 HTT (0.65) HTTKMT2ACYP2C9CYP3A4CYP2C19
SCHEMBL2399935 0.72 HTT (0.96) HTTKMT2ACYP2C9CYP3A4CYP2C19
SCHEMBL28639115 0.72 HTT (0.59) HTTCTSLCTSBCTSKMEN1
N-Piperidinobenzamide SCHEMBL696161 0.71 HTT (1.00) HTTKMT2ACYP2C9SMN1; SMN2LMNA
SCHEMBL9282775 0.71 HTT (1.00) HTTKMT2ACYP2C9SMN1; SMN2LMNA
SCHEMBL7449374 0.71 CCR3 (0.60) HTTMEN1KMT2A
SCHEMBL4630363 0.70 GNAI3 (0.37) HTTMEN1KMT2ASMN1; SMN2GAA
SCHEMBL7716857 0.68 HTT (0.69) HTTCYP2C9CYP3A4CYP2C19SMN1; SMN2
SCHEMBL1576773 0.68 CYP2D6 (0.71) HTTKMT2ACYP2C9CYP3A4CYP2C19
SCHEMBL717372 0.68 HTT (0.69) HTTCYP2C9CYP3A4CYP2C19SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1919907-A2 HETEROCYCLIC COMPOUND OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2008-05-14 EP disclosed
WO-2007026959-A2 DERIVATIVES OF 4-PIPERAZIN-1-YL-4-BENZ0 [B] THIOPHENE SUITABLE FOR THE TREATMENT OF CNS DISORDERS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2007-03-08 WO disclosed