SCHEMBL4629759

SCHEMBL4629759

O=c1[nH]cc(C2=CC=CCC2=S)c(=O)[nH]1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.40
ATAD2 Q6PL18 1/20 0.38
LMNA P02545 2/20 0.35
DPYD Q12882 4/20 0.34
MAPT P10636 2/20 0.34
GAA P10253 2/20 0.34
CYP19A1 P11511 1/20 0.34
TSHR P16473 1/20 0.34
THPO P40225 1/20 0.34
MTOR P42345 1/20 0.34
HTT P42858 1/20 0.34
HBB P68871 1/20 0.34
PMP22 Q01453 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
NT5E P21589 2/20 0.34
KDM4C Q9H3R0 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5801644 0.69 ALDH1A1 (0.64) ALDH1A1ATAD2LMNADPYDMAPT
SCHEMBL11600094 0.69
SCHEMBL8075442 0.61
SCHEMBL5146148 0.60
SCHEMBL16266667 0.60
SCHEMBL25367974 0.59 KDM3B (0.37) ALDH1A1
SCHEMBL15920864 0.59
SCHEMBL5503705 0.59 NISCH (0.37) ALDH1A1CYP19A1MTORSMN1; SMN2
SCHEMBL5612855 0.59
SCHEMBL3553811 0.59 ATAD2 (0.50) ALDH1A1ATAD2LMNADPYDMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1573000-B1 CRYSTAL STRUCTURE OF GLUTAMATE RACEMASE (MURI) ASTRAZENECA AB (SE) 2008-05-07 EP disclosed
EP-1573000-A2 CRYSTAL STRUCTURE OF GLUTAMATE RACEMASE (MURI) AstraZeneca AB (SE) 2005-09-14 EP disclosed
US-20050037478-A1 Crystal structure of glutamate racemase (MurI) ASTRAZENECA AB (SE) 2005-02-17 US disclosed
WO-2004061097-A2 CRYSTAL STRUCTURE OF GLUTAMATE RACEMASE (MURI) ASTRAZENECA AB (SE) 2004-07-22 WO disclosed