SCHEMBL4629802

SCHEMBL4629802

COc1ccc(OC)c(CC2(Nc3ccc(CC4=NCCN4)cc3)NCCN2)c1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTGIR P43119 3/20 0.49
HTR1B P28222 3/20 0.48
HTR1D P28221 5/20 0.42
ADRA2A P08913 6/20 0.39
ADRA1D P25100 4/20 0.39
ADRA1A P35348 4/20 0.39
ADRA1B P35368 4/20 0.39
ADRA2C P18825 4/20 0.39
ADRA2B P18089 3/20 0.39
TAAR1 Q96RJ0 3/20 0.38
CYP2D6 P10635 2/20 0.38
NFKB1 P19838 1/20 0.38
LMNA P02545 1/20 0.38
CYP1A2 P05177 1/20 0.38
TSHR P16473 1/20 0.38
RAD52 P43351 1/20 0.37
WDR5 P61964 2/20 0.37
GPR65 Q8IYL9 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL953504 0.77 HTR1B (0.60) PTGIRHTR1BHTR1DADRA2AADRA1D
SCHEMBL4629792 0.77 PTGIR (0.57) PTGIRHTR1BHTR1DADRA2AADRA1D
SCHEMBL4629571 0.76 TAAR1 (0.48) HTR1BHTR1DADRA2AADRA1DADRA1A
SCHEMBL9575262 0.73 PTGIR (0.83) PTGIRHTR1BHTR1DADRA2AADRA1D
SCHEMBL3169344 0.68 PTGIR (0.64) PTGIRHTR1BHTR1DADRA2AADRA1D
SCHEMBL5803714 0.67 PTGIR (1.00) PTGIRHTR1BHTR1DADRA2AADRA1D
Hydrochloric Acid SCHEMBL4692716 0.66 PTGIR (0.72) PTGIRADRA2AADRA2CADRA2BGPR65
SCHEMBL4992378 0.66 ALDH1A1 (0.61) PTGIRHTR1BHTR1DADRA2AADRA1D
SCHEMBL4687666 0.65 PTGIR (0.74) PTGIRADRA2AADRA1DADRA1AADRA1B
SCHEMBL10777223 0.64 HTR1B (0.57) PTGIRHTR1BHTR1DADRA2AADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1981497-A2 USE OF SUBSTITUTED 2-IMIDAZOLE OF IMIDAZOLINE DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 2008-10-22 EP claimed
WO-2007085557-A2 USE OF SUBSTITUTED 2-IMIDAZOLE OF IMIDAZOLINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2007-08-02 WO claimed