SCHEMBL4629792

SCHEMBL4629792

COc1ccc(OC)c(CC2=NCCN2)c1.Nc1ccc(CC2=NCCN2)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGIR P43119 2/20 0.57
HTR1B P28222 3/20 0.56
RAD52 P43351 1/20 0.54
HTR1D P28221 5/20 0.48
ADRA1A P35348 5/20 0.45
ADRA2A P08913 4/20 0.45
ADRA1D P25100 4/20 0.45
ADRA1B P35368 4/20 0.45
ADRA2C P18825 3/20 0.45
ADRA2B P18089 2/20 0.45
TAAR1 Q96RJ0 4/20 0.44
CYP2D6 P10635 2/20 0.44
NFKB1 P19838 1/20 0.44
LMNA P02545 2/20 0.44
CYP1A2 P05177 1/20 0.44
TSHR P16473 1/20 0.44
HSP90AA1 P07900 1/20 0.42
HSP90AB1 P08238 1/20 0.42
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL953504 0.89 HTR1B (0.60) PTGIRHTR1BHTR1DADRA1AADRA2A
SCHEMBL9575262 0.80 PTGIR (0.83) PTGIRHTR1BRAD52HTR1DADRA1A
SCHEMBL953972 0.78 RAD52 (0.82) PTGIRHTR1BRAD52HTR1DADRA1A
SCHEMBL4629802 0.77 PTGIR (0.49) PTGIRHTR1BRAD52HTR1DADRA1A
SCHEMBL4992378 0.76 ALDH1A1 (0.61) PTGIRHTR1BRAD52HTR1DADRA1A
SCHEMBL5803714 0.73 PTGIR (1.00) PTGIRHTR1BRAD52HTR1DADRA1A
SCHEMBL26078623 0.72 NISCH (0.58) HTR1BHTR1DADRA1AADRA2AADRA1D
SCHEMBL4629569 0.71 RAD52 (0.61) HTR1BRAD52HTR1DADRA1AADRA2A
SCHEMBL7806407 0.70 CYP19A1 (0.69) ADRA1ATAAR1IDO1DHFR
SCHEMBL26078498 0.70 HTR1B (0.55) PTGIRHTR1BHTR1DADRA1AADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1981497-A2 USE OF SUBSTITUTED 2-IMIDAZOLE OF IMIDAZOLINE DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 2008-10-22 EP claimed
WO-2007085557-A2 USE OF SUBSTITUTED 2-IMIDAZOLE OF IMIDAZOLINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2007-08-02 WO claimed