SCHEMBL4630272

SCHEMBL4630272

CC(C1=NCCN1)c1ccccc1Cl.CCC(C1=NCCN1)c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 9/20 0.50
ADRA2B P18089 9/20 0.50
ADRA2C P18825 9/20 0.50
HTR1A P08908 1/20 0.45
SLC6A4 P31645 1/20 0.45
ADRA1A P35348 1/20 0.45
OPRK1 P41145 1/20 0.45
KCNH2 Q12809 1/20 0.45
NISCH Q9Y2I1 9/20 0.45
MAOA P21397 7/20 0.45
MAOB P27338 7/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL953164 0.87 ADRA2A (0.62) ADRA2AADRA2BADRA2CHTR1ASLC6A4
SCHEMBL954219 0.84 NISCH (0.56) ADRA2AADRA2BADRA2CNISCHMAOA
SCHEMBL953759 0.77 ADRA2B (0.46) ADRA2AADRA2BADRA2CHTR1ASLC6A4
SCHEMBL954357 0.76 ADRA2A (0.44) ADRA2AADRA2BADRA2CHTR1ASLC6A4
SCHEMBL952920 0.75 ADRA2A (0.65) ADRA2AADRA2BADRA2CNISCHMAOA
SCHEMBL953349 0.73 ADRA2A (0.60) ADRA2AADRA2BADRA2CHTR1ANISCH
SCHEMBL954708 0.73 NISCH (0.45) ADRA2AADRA2BADRA2CNISCHMAOA
SCHEMBL953296 0.73 NISCH (0.53) ADRA2AADRA2BADRA2CHTR1ANISCH
SCHEMBL954868 0.73 ADRA2A (0.46) ADRA2AADRA2BADRA2CNISCHMAOA
SCHEMBL954884 0.72 NISCH (0.49) ADRA2AADRA2BADRA2CHTR1ANISCH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1981497-A2 USE OF SUBSTITUTED 2-IMIDAZOLE OF IMIDAZOLINE DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 2008-10-22 EP disclosed
WO-2007085557-A2 USE OF SUBSTITUTED 2-IMIDAZOLE OF IMIDAZOLINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2007-08-02 WO disclosed