SCHEMBL4630452

SCHEMBL4630452

CC(C)(C)OC(=O)NC1CCCCN1[C]=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSK P43235 3/20 0.48
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
BTK Q06187 2/20 0.41
GAA P10253 2/20 0.40
EPHX1 P07099 2/20 0.40
HSD11B1 P28845 2/20 0.38
CYP2C9 P11712 1/20 0.38
NFKB1 P19838 1/20 0.36
NFKB2 Q00653 1/20 0.36
RELA Q04206 1/20 0.36
JAK3 P52333 1/20 0.36
KMT2A Q03164 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
HPGD P15428 1/20 0.35
HDAC4 P56524 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
KCNA3 P22001 1/20 0.35
CTSL P07711 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL945980 0.89 CTSK (0.48) CTSKCA1CA2BTKGAA
SCHEMBL4630786 0.78 CA1 (0.36) CA1CA2GAAEPHX1HPGD
SCHEMBL5390789 0.78 CTSK (0.43) CTSKCA1CA2BTKGAA
SCHEMBL8484888 0.78 BTK (0.49) CTSKCA1CA2BTKGAA
SCHEMBL9078128 0.74 HSD17B10 (0.48) CTSKCA1CA2BTKEPHX1
SCHEMBL7017564 0.73 EPHX1 (0.40) CTSKCA1CA2BTKGAA
SCHEMBL2025019 0.73 BTK (0.50) CTSKCA1CA2BTKGAA
SCHEMBL4629917 0.73 CA1 (0.41) CA1CA2EPHX1
SCHEMBL14941684 0.72 CTSK (0.64) CTSKCA1CA2BTKGAA
SCHEMBL6687856 0.72 EPHX1 (0.42) CTSKCA1CA2BTKGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1919907-A2 HETEROCYCLIC COMPOUND OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2008-05-14 EP disclosed
WO-2007026959-A2 DERIVATIVES OF 4-PIPERAZIN-1-YL-4-BENZ0 [B] THIOPHENE SUITABLE FOR THE TREATMENT OF CNS DISORDERS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2007-03-08 WO disclosed