SCHEMBL4629917

SCHEMBL4629917

CC(=O)NC1CCCN1[C]=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.41
CA2 P00918 2/20 0.41
CA12 O43570 1/20 0.41
CA9 Q16790 1/20 0.41
ALDH1A1 P00352 2/20 0.33
KDM4E B2RXH2 2/20 0.33
EPHX2 P34913 2/20 0.32
EPHX1 P07099 1/20 0.32
ATM Q13315 1/20 0.32
FAP Q12884 3/20 0.31
PREP P48147 2/20 0.31
DPP4 P27487 1/20 0.31
PSEN1 P49768 3/20 0.30
PSEN2 P49810 3/20 0.30
APH1B Q8WW43 3/20 0.30
NCSTN Q92542 3/20 0.30
APH1A Q96BI3 3/20 0.30
PSENEN Q9NZ42 3/20 0.30
MTNR1A P48039 1/20 0.30
MTNR1B P49286 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4630786 0.95 CA1 (0.36) CA1CA2CA12CA9ALDH1A1
SCHEMBL14076271 0.75 CA1 (0.40) CA1CA2CA12CA9ALDH1A1
SCHEMBL4630168 0.74 SMN1; SMN2 (0.40) ALDH1A1MTNR1AMTNR1B
SCHEMBL8540220 0.73 DPP4 (0.41) KDM4EFAPDPP4
SCHEMBL4630452 0.73 CTSK (0.48) CA1CA2EPHX1
SCHEMBL8540218 0.73 DPP4 (0.41) KDM4EFAPDPP4
SCHEMBL6355919 0.72 CA1 (0.38) CA1CA2CA12CA9ALDH1A1
SCHEMBL6039382 0.71 LMNA (0.34) CA1CA2CA12CA9ALDH1A1
SCHEMBL3469200 0.71
SCHEMBL7451803 0.70 LMNA (0.36) DPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1919907-A2 HETEROCYCLIC COMPOUND OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2008-05-14 EP disclosed
WO-2007026959-A2 DERIVATIVES OF 4-PIPERAZIN-1-YL-4-BENZ0 [B] THIOPHENE SUITABLE FOR THE TREATMENT OF CNS DISORDERS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2007-03-08 WO disclosed