SCHEMBL4630656

SCHEMBL4630656

CCCCc1cccc(-c2ccccc2)c1[O]

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDCD1 Q15116 1/20 0.43
CD274 Q9NZQ7 1/20 0.43
NR1H2 P55055 1/20 0.42
NR1H3 Q13133 1/20 0.42
FOLH1 Q04609 1/20 0.41
PPARA Q07869 2/20 0.40
SOAT1 P35610 2/20 0.40
DPP4 P27487 1/20 0.40
BID P55957 3/20 0.40
MCL1 Q07820 3/20 0.40
BCL2L1 Q07817 2/20 0.40
BAK1 Q16611 2/20 0.40
KAT8 Q9H7Z6 2/20 0.40
PPARG P37231 1/20 0.40
EP300 Q09472 1/20 0.40
KAT2A Q92830 1/20 0.40
KAT2B Q92831 1/20 0.40
KAT5 Q92993 1/20 0.40
SAE1 Q9UBE0 1/20 0.40
LIPG Q9Y5X9 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4630157 0.95 NR1H2 (0.48) PDCD1CD274NR1H2NR1H3PPARA
SCHEMBL4630263 0.93 NR1H2 (0.50) NR1H2NR1H3PPARASOAT1BID
SCHEMBL3563200 0.89 PDCD1 (0.46) PDCD1CD274FOLH1PPARASOAT1
SCHEMBL3563149 0.83 PDCD1 (0.50) PDCD1CD274FOLH1PPARADPP4
SCHEMBL367335 0.83 DPP4 (0.52) PDCD1CD274NR1H2NR1H3FOLH1
SCHEMBL27835204 0.82 PPARA (0.48) PDCD1CD274NR1H2NR1H3FOLH1
SCHEMBL28825457 0.82 DPP4 (0.50) PDCD1CD274NR1H2NR1H3FOLH1
Ethane SCHEMBL1275986 0.82 DPP4 (0.50) PDCD1CD274NR1H2NR1H3FOLH1
SCHEMBL27424929 0.82 DPP4 (0.50) PDCD1CD274NR1H2NR1H3FOLH1
Phosphine SCHEMBL27550721 0.82 DPP4 (0.50) PDCD1CD274NR1H2NR1H3FOLH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1919907-A2 HETEROCYCLIC COMPOUND OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2008-05-14 EP disclosed
WO-2007026959-A2 DERIVATIVES OF 4-PIPERAZIN-1-YL-4-BENZ0 [B] THIOPHENE SUITABLE FOR THE TREATMENT OF CNS DISORDERS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2007-03-08 WO disclosed