SCHEMBL4631300

SCHEMBL4631300

O=C(NC1(c2ccccc2)CCNCC1)N1CCOCC1

nearest known ligand 0.58

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.58
CYP2C9 P11712 1/20 0.50
CYP2C19 P33261 1/20 0.50
SMN1; SMN2 Q16637 2/20 0.48
CYP1A2 P05177 1/20 0.47
CYP2D6 P10635 1/20 0.47
NPSR1 Q6W5P4 2/20 0.46
GAA P10253 1/20 0.46
MAPT P10636 1/20 0.46
HPGD P15428 1/20 0.46
TSHR P16473 4/20 0.43
POLB P06746 1/20 0.43
LMNA P02545 1/20 0.42
CNR1 P21554 2/20 0.42
RAB9A P51151 1/20 0.42
KDM4E B2RXH2 1/20 0.41
HSD17B10 Q99714 1/20 0.41
HTT P42858 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4630040 0.88 CYP1A2 (0.50) ALDH1A1CYP1A2CYP2D6NPSR1GAA
Benzene SCHEMBL27392883 0.88 CYP1A2 (0.50) ALDH1A1CYP1A2CYP2D6NPSR1GAA
SCHEMBL7749112 0.87 ALDH1A1 (0.49) ALDH1A1CYP2C9CYP2C19SMN1; SMN2GAA
Water SCHEMBL7749371 0.86 ALDH1A1 (0.48) ALDH1A1CYP2C9CYP2C19SMN1; SMN2GAA
Hydrochloric Acid SCHEMBL8369953 0.81 ALDH1A1 (0.58) ALDH1A1CYP2C9CYP2C19SMN1; SMN2CYP1A2
SCHEMBL7744594 0.80 CYP1A2 (0.43) ALDH1A1CYP2C19SMN1; SMN2CYP1A2CYP2D6
SCHEMBL4631302 0.77 ALDH1A1 (0.60) ALDH1A1CYP2C9CYP2C19SMN1; SMN2TSHR
SCHEMBL373284 0.77 SMN1; SMN2 (0.74) ALDH1A1CYP2C19SMN1; SMN2NPSR1TSHR
Hydrochloric Acid SCHEMBL8365023 0.77 ALDH1A1 (0.53) ALDH1A1CYP2C9CYP2C19SMN1; SMN2CYP1A2
SCHEMBL6972395 0.77 OPRM1 (0.50) ALDH1A1CYP1A2CYP2D6HPGDPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1923391-A1 Substituted heterocyclic compounds, method for preparing same and pharmaceutical compositions containing them. sanofi-aventis (FR) 2008-05-21 EP disclosed
EP-1688416-A1 Substituted heterocyclic compounds, their process of preparation and pharmaceutical compositions containing them Sanofi-Aventis (FR) 2006-08-09 EP disclosed
EP-1156049-B1 Substituted heterocyclic compounds, their process of preparation and pharmaceutical compositions containing them SANOFI AVENTIS (FR) 2005-06-01 EP disclosed
EP-1340754-A1 Substituted heterocyclic compounds, process for their preparation and pharmaceutical compositions containing them SANOFI-SYNTHELABO (FR) 2003-09-03 EP disclosed
EP-0807111-B1 SUBSTITUTED HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME SANOFI SYNTHELABO (FR) 2002-08-14 EP disclosed
EP-1156049-A1 Substituted heterocyclic compounds, their process of preparation and pharmaceutical compositions containing them SANOFI-SYNTHELABO (FR) 2001-11-21 EP disclosed
EP-0807111-A1 SUBSTITUTED HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME SANOFI (FR) 1997-11-19 EP disclosed
WO-1996023787-A1 SUBSTITUTED HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME SANOFI (FR) 1996-08-08 WO disclosed