SCHEMBL4631472

SCHEMBL4631472

Cc1cc(C=O)c(Cl)nc1C(=O)O.Cc1cnc(Cl)c(C=O)c1.O=Cc1cc(-c2ccccc2)cnc1Cl

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.36
KDM4E B2RXH2 2/20 0.36
MEN1 O00255 2/20 0.36
MAPT P10636 2/20 0.36
KMT2A Q03164 2/20 0.36
MPI P34949 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
PSMB5 P28074 1/20 0.36
MDM2 Q00987 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C19 P33261 1/20 0.35
NPSR1 Q6W5P4 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
LDHA P00338 1/20 0.34
KDR P35968 1/20 0.34
GRIN2B Q13224 2/20 0.33
DHODH Q02127 1/20 0.33
PIK3CD O00329 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2855526 0.96 CYP1A2 (0.38) ALDH1A1KDM4EMEN1MAPTKMT2A
SCHEMBL4631569 0.80 CYP1A2 (0.43) ALDH1A1KDM4EMEN1MAPTKMT2A
SCHEMBL2855346 0.79 CYP3A4 (0.51) ALDH1A1KDM4EMEN1MAPTKMT2A
SCHEMBL2847202 0.78 ALDH1A1 (0.51) ALDH1A1KDM4EMEN1MAPTKMT2A
SCHEMBL2851214 0.72 ALDH1A1 (0.47) ALDH1A1KDM4EMEN1MAPTKMT2A
SCHEMBL29954957 0.72 ALDH1A1 (0.47) ALDH1A1KDM4EMEN1MAPTKMT2A
SCHEMBL2849385 0.69 CYP1A2 (0.53) ALDH1A1KDM4EMEN1MAPTKMT2A
SCHEMBL11153472 0.66 ERN1 (0.51) ALDH1A1KDM4EMAPTKMT2ASMN1; SMN2
SCHEMBL22445783 0.65 CYP1A2 (0.47) ALDH1A1KDM4EMEN1MAPTKMT2A
SCHEMBL2849379 0.65 ALDH1A1 (0.56) ALDH1A1KDM4EMAPTSMN1; SMN2PSMB5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1924558-A1 AN ANTIMALARIAL BAYLIS-HILLMAN ADDUCTS AND A PROCESS FOR THE PREPARATION THEREOF COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2008-05-28 EP claimed
WO-2007032016-A1 AN ANTIMALARIAL BAYLIS-HILLMAN ADDUCTS AND A PROCESS FOR THE PREPARATION THEREOF COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2007-03-22 WO claimed