SCHEMBL4632644

SCHEMBL4632644

CC(C)(C)NC(=O)c1cccnc1CC(=O)C(Cc1ccc(Cl)cc1)NC(=O)O

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 3/20 0.42
ITGA4 P13612 3/20 0.42
SMN1; SMN2 Q16637 1/20 0.40
CAPN1 P07384 2/20 0.38
CNR1 P21554 2/20 0.38
CNR2 P34972 1/20 0.38
KMT2A Q03164 3/20 0.37
MEN1 O00255 2/20 0.37
GPR132 Q9UNW8 1/20 0.37
EGLN1 Q9GZT9 1/20 0.36
SCN9A Q15858 1/20 0.36
USP30 Q70CQ3 2/20 0.35
P2RX7 Q99572 1/20 0.35
MAPT P10636 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
ITGB7 P26010 1/20 0.35
PPARG P37231 1/20 0.35
WDR5 P61964 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL278005 0.89 SCN9A (0.45) KMT2AMEN1SCN9AMAPTNPSR1
SCHEMBL4667376 0.85 ANO1 (0.45) SMN1; SMN2CAPN1KMT2AMAPT
SCHEMBL4837212 0.85 ANO1 (0.41) SMN1; SMN2P2RX7
SCHEMBL4632200 0.83 SMN1; SMN2 (0.43) SMN1; SMN2CAPN1KMT2AMEN1MAPT
SCHEMBL269012 0.77 PTPN1 (0.42) SCN9A
SCHEMBL269828 0.77 SMN1; SMN2 (0.40) SMN1; SMN2CAPN1CNR1CNR2KMT2A
SCHEMBL268438 0.77 SCN9A (0.40) SMN1; SMN2SCN9AMAPT
SCHEMBL277711 0.76 ACE (0.43) KMT2ASCN9AMAPTNPSR1
Hydrochloric Acid SCHEMBL268993 0.76 SMN1; SMN2 (0.39) SMN1; SMN2CAPN1CNR1CNR2KMT2A
SCHEMBL268932 0.76 ANO1 (0.43) SCN9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1912946-A1 PYRIDINE DERIVATIVES AS DIPEPTEDYL PEPTIDASE INHIBITORS Eli Lilly and Company (US) 2008-04-23 EP disclosed
WO-2007015767-A1 PYRIDINE DERIVATIVES AS DIPEPTEDYL PEPTIDASE INHIBITORS ELI LILLY AND COMPANY (US) 2007-02-08 WO disclosed