SCHEMBL463285

SCHEMBL463285

COc1cccc(Nc2cc(NCC(C)(C)O)c3ncc(-c4ccc(C(N)=O)c(C)c4C4CC4)n3n2)c1

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PDE4D Q08499 10/20 0.43
PDE4B Q07343 9/20 0.43
PDE4A P27815 7/20 0.43
PDE4C Q08493 7/20 0.43
TYK2 P29597 7/20 0.42
TTK P33981 1/20 0.40
SYK P43405 1/20 0.37
CNR2 P34972 1/20 0.37
CCNE1 P24864 1/20 0.36
CDK2 P24941 1/20 0.36
FLT3 P36888 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL462124 0.80 TTK (0.49) TTK
SCHEMBL463247 0.80 TTK (0.47) TTK
SCHEMBL461988 0.80 TTK (0.40) PDE4DTYK2TTK
SCHEMBL456319 0.79 TTK (0.57) TTK
SCHEMBL12467108 0.76 TTK (0.36) TTKSYKFLT3
SCHEMBL456965 0.76 ERN1 (0.40) TTKFLT3
SCHEMBL462359 0.75 TTK (0.42) TTKSYK
SCHEMBL457467 0.71 TTK (0.40) TTK
SCHEMBL457970 0.71 TTK (0.44) TTK
SCHEMBL9942420 0.71 TTK (0.44) TTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2614063-A1 SUBSTITUTED IMIDAZOPYRIDAZINES Bayer Intellectual Property GmbH (DE) 2013-07-17 EP disclosed
WO-2012032031-A1 SUBSTITUTED IMIDAZOPYRIDAZINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2012-03-15 WO disclosed