SCHEMBL4633571

SCHEMBL4633571

COC(=O)CCc1ccc(OCCOc2c(C(=O)O)sc3ccccc23)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CXCR2 P25025 1/20 0.55
LTA4H P09960 2/20 0.45
BCL2 P10415 1/20 0.44
BCL2L1 Q07817 1/20 0.44
MCL1 Q07820 1/20 0.44
BAD Q92934 1/20 0.44
TSHR P16473 1/20 0.44
ALDH1A1 P00352 2/20 0.43
LMNA P02545 2/20 0.43
FFAR1 O14842 3/20 0.43
PPARG P37231 1/20 0.43
EDNRA P25101 1/20 0.42
MAPT P10636 1/20 0.42
RXFP1 Q9HBX9 1/20 0.42
TP53 P04637 1/20 0.42
CASP3 P42574 1/20 0.42
CASP7 P55210 1/20 0.42
SENP5 Q96HI0 1/20 0.42
SENP2 Q9HC62 1/20 0.42
SENP1 Q9P0U3 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4603385 0.91 CXCR2 (0.53) CXCR2LTA4HTSHRALDH1A1LMNA
SCHEMBL4635068 0.88 LMNA (0.51) CXCR2ALDH1A1LMNAMAPTRXFP1
SCHEMBL4604985 0.83 CXCR2 (0.54) CXCR2LMNAFFAR1PPARGMAPT
SCHEMBL4633866 0.83 CXCR2 (0.67) CXCR2BCL2BCL2L1MCL1BAD
SCHEMBL4635016 0.82 CXCR2 (0.43) CXCR2LTA4HALDH1A1LMNAPPARG
SCHEMBL4828979 0.80 CXCR2 (0.57) CXCR2LMNAFFAR1PPARG
SCHEMBL4633030 0.80 CXCR2 (0.52) CXCR2LMNAFFAR1PPARG
SCHEMBL13932451 0.80 FFAR1 (0.60) LTA4HLMNAFFAR1PPARGMAPT
SCHEMBL4603395 0.80 FFAR1 (0.53) CXCR2LMNAFFAR1
SCHEMBL4635058 0.79 CXCR2 (0.58) CXCR2BCL2BCL2L1MCL1BAD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1685121-B1 ANTIDIABETIC COMPOUNDS COMPRISING BENZOTHIOPHENE DERIVATIVES MERCK PATENT GMBH (DE) 2008-06-11 EP claimed