SCHEMBL4633952

SCHEMBL4633952

CCOC(=O)Oc1sc2ccccc2c1OCCOc1ccc(C#N)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CXCR2 P25025 1/20 0.44
ALDH1A1 P00352 3/20 0.43
KMT2A Q03164 2/20 0.43
LMNA P02545 2/20 0.43
MAPT P10636 3/20 0.43
NOD2 Q9HC29 1/20 0.42
CYP11B1 P15538 1/20 0.40
CYP11B2 P19099 1/20 0.40
GAA P10253 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
HRH2 P25021 1/20 0.39
HRH1 P35367 1/20 0.39
HRH3 Q9Y5N1 1/20 0.39
GABRP O00591 1/20 0.39
GABRD O14764 1/20 0.39
GABRA1 P14867 1/20 0.39
GABRB1 P18505 1/20 0.39
GABRG2 P18507 1/20 0.39
GABRB3 P28472 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4635043 0.89 CXCR2 (0.55) CXCR2ALDH1A1KMT2ALMNAMAPT
SCHEMBL4632905 0.88 ALDH1A1 (0.43) ALDH1A1KMT2ALMNAMAPTNOD2
SCHEMBL4633878 0.87 CXCR2 (0.46) CXCR2ALDH1A1KMT2ALMNAMAPT
SCHEMBL4633540 0.86 CXCR2 (0.51) CXCR2ALDH1A1KMT2ALMNAMAPT
SCHEMBL4633874 0.85 ALDH1A1 (0.56) CXCR2ALDH1A1KMT2ALMNAMAPT
SCHEMBL4635016 0.81 CXCR2 (0.43) CXCR2ALDH1A1KMT2ALMNAMAPT
SCHEMBL4632951 0.81 FFAR1 (0.45) ALDH1A1KMT2ALMNAMAPTNOD2
SCHEMBL4633609 0.80 LMNA (0.54) CXCR2ALDH1A1KMT2ALMNAMAPT
SCHEMBL4633576 0.79 KMT2A (0.50) CXCR2ALDH1A1KMT2ALMNAMAPT
SCHEMBL4634428 0.79 ALDH1A1 (0.43) ALDH1A1KMT2ALMNAMAPTNOD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1685121-B1 ANTIDIABETIC COMPOUNDS COMPRISING BENZOTHIOPHENE DERIVATIVES MERCK PATENT GMBH (DE) 2008-06-11 EP claimed