SCHEMBL4634183

SCHEMBL4634183

[2H]CN(c1c(C)cccc1C)c1cc(C(=O)N(C)C)cc2c1nc(C)n2C

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
GAA P10253 1/20 0.35
PABPC1 P11940 1/20 0.35
HPGD P15428 1/20 0.35
CASP1 P29466 1/20 0.35
HTT P42858 1/20 0.35
HSD17B10 Q99714 1/20 0.35
CYP1A2 P05177 2/20 0.32
CYP3A4 P08684 2/20 0.32
CYP2C9 P11712 2/20 0.32
CYP2C19 P33261 2/20 0.32
CYP2D6 P10635 1/20 0.32
BRD4 O60885 1/20 0.32
RORC P51449 1/20 0.32
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
F10 P00742 1/20 0.31
TGFBR1 P36897 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4632998 0.94 KDM4E (0.35) KDM4EALDH1A1GAAPABPC1HPGD
SCHEMBL4633218 0.88 KDM4E (0.33) KDM4EALDH1A1GAAPABPC1HPGD
SCHEMBL4634190 0.83 SLC22A12 (0.34) ALDH1A1GAAHPGDHSD17B10CYP1A2
SCHEMBL4632933 0.78 SMN1; SMN2 (0.37) KDM4EALDH1A1GAAPABPC1HPGD
SCHEMBL5901177 0.78 KDM4E (0.30) KDM4EALDH1A1GAAPABPC1HPGD
SCHEMBL3555267 0.72 ALDH1A1 (0.34) KDM4EALDH1A1GAAPABPC1HPGD
SCHEMBL5901876 0.72 CYP3A4 (0.39) KDM4EALDH1A1GAAPABPC1HPGD
SCHEMBL4592754 0.72 CYP3A4 (0.61) KDM4EALDH1A1GAAPABPC1HPGD
SCHEMBL4777017 0.71 NPC1 (0.34) KDM4EALDH1A1GAAPABPC1HPGD
SCHEMBL4592596 0.71 MAP4K1 (0.36) KDM4EALDH1A1GAAPABPC1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1926714-A1 ISOTOPICALLY SUBSTITUTED BENZIMIDAZOLE DERIVATIVES Nycomed GmbH (DE) 2008-06-04 EP claimed
WO-2007023135-A1 ISOTOPICALLY SUBSTITUTED BENZIMIDAZOLE DERIVATIVES NYCOMED GMBH (DE) 2007-03-01 WO claimed
EP-1926714-A1 ISOTOPICALLY SUBSTITUTED BENZIMIDAZOLE DERIVATIVES Nycomed GmbH (DE) 2008-06-04 EP disclosed
WO-2007023135-A1 ISOTOPICALLY SUBSTITUTED BENZIMIDAZOLE DERIVATIVES NYCOMED GMBH (DE) 2007-03-01 WO disclosed