SCHEMBL4635252

SCHEMBL4635252

O=c1[nH]cnc2nc(NC3CCNCC3)n(Cc3ccc(F)cc3)c12

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 3/20 0.57
NR4A2 P43354 2/20 0.57
SOS1 Q07889 1/20 0.44
SSTR5 P35346 5/20 0.41
MPO P05164 1/20 0.40
TPO P07202 1/20 0.40
MEN1 O00255 1/20 0.39
POLB P06746 1/20 0.39
RAB9A P51151 1/20 0.39
KMT2A Q03164 1/20 0.39
BRDT Q58F21 1/20 0.39
ALDH1A1 P00352 2/20 0.38
LMNA P02545 1/20 0.38
GAA P10253 1/20 0.38
HSD17B10 Q99714 2/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CASP1 P29466 1/20 0.38
CASP7 P55210 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4635524 0.88 SSTR5 (0.44) KCNH2NR4A2SSTR5MEN1POLB
SCHEMBL3970572 0.81 KCNH2 (0.42) KCNH2NR4A2SOS1MPOTPO
SCHEMBL3971456 0.80 HTR6 (0.39) KCNH2NR4A2SOS1MPOTPO
Bromide SCHEMBL9564852 0.80 KCNH2 (0.57) KCNH2NR4A2SOS1SSTR5MEN1
Bromide SCHEMBL9699462 0.76 KCNH2 (0.72) KCNH2NR4A2SOS1SSTR5MEN1
Hydrochloric Acid SCHEMBL9630081 0.73 KCNH2 (0.67) KCNH2NR4A2SOS1SSTR5MEN1
Tecastemizole SCHEMBL18200 0.72 KCNH2 (1.00) KCNH2NR4A2SOS1SSTR5MEN1
Tecastemizole SCHEMBL9698437 0.72 KCNH2 (0.98) KCNH2NR4A2SOS1SSTR5MEN1
Bromide SCHEMBL11304724 0.72 KCNH2 (0.78) KCNH2NR4A2SOS1SSTR5MEN1
Tecastemizole SCHEMBL11278980 0.72 KCNH2 (0.98) KCNH2NR4A2SOS1SSTR5MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1532150-B1 NOVEL PURINE DERIVATIVES, PRODUCTION AND USE THEREOF AS MEDICAMENTS BOEHRINGER INGELHEIM PHARMA (DE) 2008-06-11 EP claimed