SCHEMBL4635855

SCHEMBL4635855

Cc1c(Sc2ccc(S(C)(=O)=O)cc2F)c2cc(Cl)ccn2c1CC(=O)O

nearest known ligand 0.53

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 14/20 0.53
TBXA2R P21731 1/20 0.40
PTGS2 P35354 4/20 0.38
PTGS1 P23219 2/20 0.38
PTGDR Q13258 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4635635 0.89 PTGDR2 (0.44) PTGDR2TBXA2RPTGS2PTGS1
SCHEMBL4635553 0.85 PTGDR2 (0.48) PTGDR2
SCHEMBL27743072 0.85 PTGDR2 (0.42) PTGDR2TBXA2RPTGS2PTGS1
SCHEMBL4635352 0.79 PTGS2 (0.40) PTGDR2TBXA2RPTGS2PTGS1PTGDR
SCHEMBL27743074 0.78 PTGDR2 (0.40) PTGDR2TBXA2RPTGS2PTGS1
SCHEMBL4635776 0.75 PTGDR2 (0.39) PTGDR2PTGS2PTGS1PTGDR
SCHEMBL4636153 0.74 L3MBTL1 (0.41) PTGDR2PTGS2
SCHEMBL4779100 0.73 TSHR (0.40) PTGDR2
SCHEMBL4636887 0.73 PTGDR2 (0.43) PTGDR2TBXA2RPTGS2PTGS1PTGDR
SCHEMBL4635707 0.71 PTGDR2 (0.43) PTGDR2PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080306109-A1 Indolizine Derivatives as Ligands of the Crth2 Receptor ARGENTA DISCOVERY LIMITED (GB) 2008-12-11 US disclosed
US-20080306109-A1 Indolizine Derivatives as Ligands of the Crth2 Receptor ARGENTA DISCOVERY LIMITED (GB) 2008-12-11 US disclosed
US-20080306109-A1 Indolizine Derivatives as Ligands of the Crth2 Receptor ARGENTA DISCOVERY LIMITED (GB) 2008-12-11 US disclosed
EP-1931663-A1 IMDOLIZINE DERIVATIVES AS LIGANDS OF THE CRTH2 RECEPTOR Argenta Discovery Limited (GB) 2008-06-18 EP disclosed
WO-2007031747-A1 IMDOLIZINE DERIVATIVES AS LIGANDS OF THE CRTH2 RECEPTOR ARGENTA DISCOVERY LIMITED (GB) 2007-03-22 WO disclosed
WO-2007031747-A1 IMDOLIZINE DERIVATIVES AS LIGANDS OF THE CRTH2 RECEPTOR ARGENTA DISCOVERY LIMITED (GB) 2007-03-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080306109-A1 Indolizine Derivatives as Ligands of the Crth2 Receptor HRH4, HRH2, HRH3 PTGDR2 293/4885TBXA2R 274/4885PTGS2 896/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.