SCHEMBL4636723

SCHEMBL4636723

CCn1c(=O)c2c(nc(C#Cc3cccc(F)c3)n2C)n(CC)c1=O

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 4/20 0.47
ADORA2A P29274 4/20 0.46
ADORA2B P29275 4/20 0.45
HTR1A P08908 1/20 0.43
ADORA3 P0DMS8 1/20 0.43
CYP2C9 P11712 1/20 0.43
MAOB P27338 1/20 0.43
PDE4A P27815 1/20 0.43
PDE4D Q08499 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4636158 0.88 ADORA1 (0.48) ADORA1ADORA2AADORA2BHTR1AADORA3
SCHEMBL4636795 0.87 ADORA1 (0.47) ADORA1ADORA2AADORA2BHTR1AADORA3
SCHEMBL4637338 0.86 ADORA2A (0.61) ADORA1ADORA2AADORA2BHTR1AADORA3
SCHEMBL4636181 0.85 ADORA2A (0.55) ADORA1ADORA2AADORA2BHTR1AADORA3
SCHEMBL2534038 0.82 ADORA2A (0.47) ADORA1ADORA2AADORA2BMAOB
SCHEMBL4636001 0.81 MAOA (0.43) ADORA1MAOB
SCHEMBL2542959 0.81 ADORA2A (0.43) ADORA1ADORA2AADORA2B
SCHEMBL4636790 0.80 MAOB (0.47) ADORA2AADORA2BMAOB
SCHEMBL4637336 0.80 ADORA2A (0.60) ADORA1ADORA2AADORA2BHTR1AADORA3
SCHEMBL2542620 0.80 MAOB (0.42) ADORA1ADORA2AADORA2BMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1939197-A1 8-ethinylxanthine derivatives as selective A2A receptor antagonists SCHWARZ PHARMA AG (DE) 2008-07-02 EP disclosed