SCHEMBL4637264

SCHEMBL4637264

CCn1c(=O)c2c(nc(C#Cc3cccc(OC)c3)n2C)n(C)c1=O

nearest known ligand 0.57

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAOB P27338 5/20 0.47
ADORA2A P29274 1/20 0.47
MAOA P21397 3/20 0.47
PKM P14618 1/20 0.47
MAPT P10636 1/20 0.46
ADORA1 P30542 2/20 0.46
NCOA1 Q15788 1/20 0.45
NCOA3 Q9Y6Q9 1/20 0.45
ADORA3 P0DMS8 2/20 0.44
MEN1 O00255 1/20 0.44
ALDH1A1 P00352 1/20 0.44
KMT2A Q03164 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
HIF1A Q16665 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4636181 0.94 ADORA2A (0.55) MAOBADORA2AADORA1ADORA3
SCHEMBL2537627 0.89 ADORA1 (0.57) MAOBADORA2AADORA1
SCHEMBL4636778 0.88 ADORA2B (0.51) MAOBMAOAPKMMAPTADORA3
SCHEMBL4636116 0.88 MAOB (0.57) MAOBMAOAPKMNCOA1NCOA3
SCHEMBL2538825 0.86 ADORA1 (0.53) MAOBADORA2AADORA1ADORA3
SCHEMBL4635978 0.86 ADORA1 (0.55) MAOBADORA2AADORA1ADORA3
SCHEMBL4636001 0.86 MAOA (0.43) MAOBMAOAPKMMAPTADORA1
SCHEMBL4636790 0.85 MAOB (0.47) MAOBADORA2AMAOAALDH1A1HIF1A
SCHEMBL2548492 0.83 ADORA1 (0.57) MAOBADORA2AADORA1ADORA3
SCHEMBL2539378 0.83 ADORA1 (0.56) MAOBADORA2AADORA1ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1939197-A1 8-ethinylxanthine derivatives as selective A2A receptor antagonists SCHWARZ PHARMA AG (DE) 2008-07-02 EP disclosed