SCHEMBL4637428

SCHEMBL4637428

CCS(=O)(=O)N1CCC(NC(=O)OC(C)(C)C)CC1

nearest known ligand 0.55

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.55
CTSK P43235 2/20 0.52
GAA P10253 1/20 0.51
ALDH1A1 P00352 1/20 0.50
EPHX2 P34913 2/20 0.47
CYP2C9 P11712 1/20 0.47
HSD11B1 P28845 1/20 0.47
BRD4 O60885 2/20 0.47
BTK Q06187 1/20 0.46
KCNA3 P22001 1/20 0.46
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
CKS1B P61024 1/20 0.45
SKP1 P63208 1/20 0.45
SKP2 Q13309 1/20 0.45
SMYD3 Q9H7B4 1/20 0.44
NAMPT P43490 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14417786 0.92 ALDH1A1 (0.54) TSHRL3MBTL1CTSKGAAALDH1A1
SCHEMBL19863558 0.88 EPHX2 (0.52) TSHRL3MBTL1CTSKGAAEPHX2
SCHEMBL17557565 0.88 CTSK (0.47) TSHRL3MBTL1CTSKGAAALDH1A1
SCHEMBL30761942 0.86 TSHR (0.48) TSHRL3MBTL1CTSKGAAEPHX2
SCHEMBL25123847 0.86 CTSK (0.54) CTSKGAAEPHX2CYP2C9HSD11B1
SCHEMBL17591811 0.86 CTSK (0.54) L3MBTL1CTSKGAAEPHX2CYP2C9
SCHEMBL3841283 0.86 CTSK (0.54) CTSKALDH1A1EPHX2CYP2C9HSD11B1
SCHEMBL24572246 0.85 EPHX2 (0.46) TSHRL3MBTL1CTSKALDH1A1EPHX2
SCHEMBL23973912 0.85 CTSK (0.52) CTSKEPHX2CYP2C9HSD11B1BRD4
SCHEMBL21841177 0.85 CTSK (0.52) CTSKGAAEPHX2CYP2C9HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230174488-A1 SARS-COV-2 INHIBITORS HAVING COVALENT MODIFICATIONS FOR TREATING CORONAVIRUS INFECTIONS INSILICO MEDICINE IP LIMITED (HK) 2023-06-08 US disclosed
WO-2021219089-A1 SARS-COV-2 INHIBITORS HAVING COVALENT MODIFICATIONS FOR TREATING CORONAVIRUS INFECTIONS INSILICO MEDICINE IP LIMITED (CN) 2021-11-04 WO disclosed
WO-2021003314-A1 HETEROCYCLIC COMPOUNDS AS KINASE INHIBITORS NUVATION BIO INC. (US) 2021-01-07 WO disclosed
EP-1951678-A1 PYRAZOLE COMPOUNDS HAVING CANNABINOID RECEPTOR (CB1) ANTAGONIZING ACTIVITY Mitsubishi Tanabe Pharma Corporation (JP) 2008-08-06 EP disclosed
US-7268150-B2 2-cyano-4-fluoropyrrolidine derivative or its salt YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 2007-09-11 US disclosed
WO-2007046550-A1 PYRAZOLE COMPOUNDS HAVING CANNABINOID RECEPTOR (CB1) ANTAGONIZING ACTIVITY MITSUBISHI TANABE PHARMA CORPORATION (JP) 2007-04-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230174488-A1 SARS-COV-2 INHIBITORS HAVING COVALENT MODIFICATIONS FOR TREATING CORONAVIRUS INFECTIONS ACE2, SARS1, ACE TSHR 4532/4885L3MBTL1 2882/4885CTSK 158/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.