SCHEMBL4637784

SCHEMBL4637784

O=C(c1nnn(Cc2cc(C(F)(F)F)cc(C(F)(F)F)c2)c1-c1cccnc1)c1c(CCOC2CCCCO2)noc1-c1ccccc1Cl

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 1/20 0.37
MET P08581 1/20 0.33
CRHR1 P34998 1/20 0.32
CYP11B1 P15538 1/20 0.32
CYP11B2 P19099 1/20 0.32
GPBAR1 Q8TDU6 4/20 0.32
ALDH1A1 P00352 1/20 0.31
TSHR P16473 1/20 0.31
PDE8B O95263 1/20 0.31
KDM4C Q9H3R0 1/20 0.30
TACR1 P25103 2/20 0.30
RORC P51449 1/20 0.30
SRPK1 Q96SB4 1/20 0.30
CFTR P13569 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4637728 0.95 IDH1 (0.37) IDH1METCRHR1GPBAR1ALDH1A1
SCHEMBL4638809 0.94 ALDH1A1 (0.36) ALDH1A1TSHRKDM4CRORC
SCHEMBL4638885 0.93 TRPV1 (0.32) IDH1METGPBAR1ALDH1A1TSHR
SCHEMBL4638641 0.90 IDH1 (0.41) IDH1METCRHR1ALDH1A1TSHR
SCHEMBL4638099 0.90 IDH1 (0.36) IDH1CRHR1CYP11B1CYP11B2ALDH1A1
SCHEMBL4639054 0.88 ALDH1A1 (0.36) ALDH1A1TSHRTACR1RORCCFTR
SCHEMBL4638821 0.88 TACR1 (0.32) IDH1GPBAR1ALDH1A1TSHRTACR1
SCHEMBL4637757 0.87 ALDH1A1 (0.33) IDH1METALDH1A1TSHRPDE8B
SCHEMBL4708380 0.87 IDH1 (0.42) IDH1CRHR1GPBAR1ALDH1A1TSHR
SCHEMBL4638945 0.86 IDH1 (0.35) IDH1CRHR1PDE8BRORCCFTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501808-B1 TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-07-02 EP disclosed
EP-1501809-B1 TRIAZOLE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-01-16 EP disclosed