SCHEMBL4638945

SCHEMBL4638945

O=C(c1nnn(Cc2cc(C(F)(F)F)ccc2C(F)(F)F)c1-c1cccnc1)c1c(COC2CCCCO2)noc1-c1ccccc1Cl

nearest known ligand 0.35

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 1/20 0.35
CFTR P13569 3/20 0.33
RORC P51449 2/20 0.32
CRHR1 P34998 1/20 0.32
RET P07949 2/20 0.31
PDE8B O95263 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4638641 0.92 IDH1 (0.41) IDH1CFTRRORCCRHR1PDE8B
SCHEMBL4638099 0.91 IDH1 (0.36) IDH1CFTRRORCCRHR1
SCHEMBL4637728 0.91 IDH1 (0.37) IDH1CFTRRORCCRHR1PDE8B
SCHEMBL4637757 0.87 ALDH1A1 (0.33) IDH1PDE8B
SCHEMBL4638502 0.86 CDK9 (0.34) IDH1PDE8B
SCHEMBL4637784 0.86 IDH1 (0.37) IDH1CFTRRORCCRHR1PDE8B
SCHEMBL4639054 0.85 ALDH1A1 (0.36) CFTRRORC
SCHEMBL4638821 0.84 TACR1 (0.32) IDH1CFTRRORC
SCHEMBL4639447 0.84 IDH1 (0.35) IDH1CFTRRORCCRHR1PDE8B
SCHEMBL4639496 0.82 CFTR (0.32) CFTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501808-B1 TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-07-02 EP disclosed