SCHEMBL4637824

SCHEMBL4637824

O=C(C#Cc1ccccc1F)c1nnn(Cc2cc(C(F)(F)F)cc(C(F)(F)F)c2)c1-c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.44
GAA P10253 1/20 0.44
CYP19A1 P11511 5/20 0.41
TSHR P16473 1/20 0.41
POLB P06746 2/20 0.39
GRM2 Q14416 2/20 0.39
ADORA3 P0DMS8 2/20 0.37
AKR1C3 P42330 1/20 0.35
AKR1C2 P52895 1/20 0.35
PTGER4 P35408 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
RORC P51449 1/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.34
TACR1 P25103 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4638053 0.90 ALDH1A1 (0.44) ALDH1A1GAACYP19A1TSHRPOLB
SCHEMBL4637826 0.88 ALDH1A1 (0.47) ALDH1A1GAACYP19A1TSHRPOLB
SCHEMBL4638482 0.87 ALDH1A1 (0.44) ALDH1A1GAACYP19A1TSHRPOLB
SCHEMBL4637775 0.85 POLB (0.45) ALDH1A1GAACYP19A1TSHRPOLB
SCHEMBL4637813 0.84 IDH1 (0.39) ALDH1A1GAACYP19A1TSHRGRM2
SCHEMBL4638563 0.83 ALDH1A1 (0.47) ALDH1A1GAACYP19A1TSHRPOLB
SCHEMBL4707915 0.82 IDH1 (0.48) ALDH1A1GAACYP19A1TSHRGRM2
SCHEMBL4638473 0.81 ALDH1A1 (0.65) ALDH1A1GAACYP19A1TSHRPOLB
SCHEMBL4637949 0.81 IDH1 (0.39) ALDH1A1GAACYP19A1TSHRGRM2
SCHEMBL4637820 0.81 GAA (0.40) ALDH1A1GAACYP19A1TSHRPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501808-B1 TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-07-02 EP disclosed