SCHEMBL4637775

SCHEMBL4637775

O=C(C#Cc1cccc(C(F)(F)F)c1)c1nnn(Cc2cc(C(F)(F)F)cc(C(F)(F)F)c2)c1-c1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.45
ALDH1A1 P00352 3/20 0.44
GAA P10253 1/20 0.44
CYP19A1 P11511 2/20 0.41
TSHR P16473 1/20 0.41
AKR1C3 P42330 1/20 0.41
AKR1C2 P52895 1/20 0.41
FFAR1 O14842 1/20 0.41
ADORA3 P0DMS8 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
PTGER4 P35408 1/20 0.40
GRIN1 Q05586 1/20 0.39
GRIN2B Q13224 1/20 0.39
TP53 P04637 2/20 0.39
MAPT P10636 3/20 0.39
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
LMNA P02545 1/20 0.39
KMT2A Q03164 1/20 0.39
GRM2 Q14416 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4637826 0.94 ALDH1A1 (0.47) POLBALDH1A1GAACYP19A1TSHR
SCHEMBL4638482 0.89 ALDH1A1 (0.44) POLBALDH1A1GAACYP19A1TSHR
SCHEMBL4637824 0.85 ALDH1A1 (0.44) POLBALDH1A1GAACYP19A1TSHR
SCHEMBL4638053 0.84 ALDH1A1 (0.44) POLBALDH1A1GAACYP19A1TSHR
SCHEMBL4638563 0.83 ALDH1A1 (0.47) POLBALDH1A1GAACYP19A1TSHR
SCHEMBL4638473 0.81 ALDH1A1 (0.65) POLBALDH1A1GAACYP19A1TSHR
SCHEMBL4637770 0.81 ADORA3 (0.46) POLBALDH1A1GAAAKR1C3AKR1C2
SCHEMBL4706776 0.81 ALDH1A1 (0.54) POLBALDH1A1GAACYP19A1TSHR
SCHEMBL4638500 0.80 POLB (0.41) POLBALDH1A1GAATSHRAKR1C3
SCHEMBL4637822 0.79 ALDH1A1 (0.43) POLBALDH1A1GAACYP19A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501808-B1 TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-07-02 EP disclosed