SCHEMBL4637835

SCHEMBL4637835

O=C(c1nnn(Cc2cc(C(F)(F)F)cc(C(F)(F)F)c2)c1-c1ccccc1)c1c(-c2ccccc2Cl)nnn1CCO

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.43
TSHR P16473 1/20 0.43
GRM2 Q14416 2/20 0.41
GAA P10253 1/20 0.40
CYP19A1 P11511 4/20 0.39
PTGER4 P35408 2/20 0.38
TACR1 P25103 2/20 0.36
IDO1 P14902 2/20 0.36
TDO2 P48775 2/20 0.36
AKR1C3 P42330 1/20 0.35
AKR1C2 P52895 1/20 0.35
ADORA3 P0DMS8 1/20 0.35
PTGES O14684 1/20 0.35
ALOX5 P09917 1/20 0.35
POLB P06746 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4638479 0.90 ALDH1A1 (0.46) ALDH1A1TSHRGRM2GAACYP19A1
SCHEMBL6230808 0.89 ALDH1A1 (0.43) ALDH1A1TSHRGRM2GAACYP19A1
SCHEMBL4638565 0.87 ALDH1A1 (0.43) ALDH1A1TSHRGRM2GAACYP19A1
SCHEMBL4639402 0.87 ALDH1A1 (0.40) ALDH1A1TSHRGRM2GAACYP19A1
SCHEMBL4705766 0.84 ALDH1A1 (0.37) ALDH1A1TSHRGRM2GAACYP19A1
SCHEMBL4638919 0.83 TACR1 (0.48) ALDH1A1TSHRGRM2GAACYP19A1
SCHEMBL4705903 0.82 IDH1 (0.44) ALDH1A1TSHRGRM2PTGER4
SCHEMBL14587206 0.82 ALDH1A1 (0.47) ALDH1A1TSHRGRM2GAACYP19A1
SCHEMBL4706457 0.81 ALDH1A1 (0.44) ALDH1A1TSHRGRM2GAACYP19A1
SCHEMBL4637956 0.80 ALDH1A1 (0.46) ALDH1A1TSHRGRM2GAACYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501808-B1 TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-07-02 EP disclosed
EP-1501808-B1 TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-07-02 EP disclosed
US-7179804-B2 Tachykinin receptor antagonists ELI LILLY AND COMPANY (US) 2007-02-20 US disclosed
EP-1501808-A1 TACHYKININ RECEPTOR ANTAGONISTS ELI LILLY AND COMPANY (US) 2005-02-02 EP disclosed
WO-2003091227-A1 TACHYKININ RECEPTOR ANTAGONISTS ELI LILLY AND COMPANY (US) 2003-11-06 WO disclosed