SCHEMBL4637844

SCHEMBL4637844

ON=Cc1ccncc1Cl

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.42
CCNT1 O60563 1/20 0.42
CDK9 P50750 1/20 0.42
HASPIN Q8TF76 1/20 0.42
HTT P42858 2/20 0.39
CDK5 Q00535 1/20 0.39
CDK5R1 Q15078 1/20 0.39
GSK3A P49840 1/20 0.36
GSK3B P49841 1/20 0.36
CYP2A6 P11509 3/20 0.36
CYP3A4 P08684 2/20 0.36
TP53 P04637 1/20 0.35
HPGD P15428 2/20 0.35
ACHE P22303 4/20 0.35
ALDH1A1 P00352 1/20 0.34
NFE2L2 Q16236 1/20 0.34
TSHR P16473 1/20 0.33
KDM4E B2RXH2 1/20 0.33
KMT2A Q03164 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4637840 1.00 GAA (0.42) GAACCNT1CDK9HASPINHTT
SCHEMBL1982834 0.86 CCNT1 (0.43) GAACCNT1CDK9HASPINHTT
SCHEMBL1982833 0.86 CCNT1 (0.43) GAACCNT1CDK9HASPINHTT
SCHEMBL25320343 0.78 CCNT1 (0.43) GAACCNT1CDK9HASPINHTT
SCHEMBL4637787 0.77 GAA (0.39) GAAHTTCDK5CDK5R1GSK3B
SCHEMBL28657657 0.77 GRIN2D (0.60) TSHRKMT2AL3MBTL1
SCHEMBL15741494 0.76
SCHEMBL6069581 0.76 CCNT1 (0.42) GAACCNT1CDK9HASPINHTT
SCHEMBL6069584 0.76 CCNT1 (0.42) GAACCNT1CDK9HASPINHTT
SCHEMBL4764878 0.76 CCNC (0.50) GAACCNT1CDK9HASPINHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501808-B1 TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-07-02 EP disclosed
CN-1313450-C Tachykinin receptor antagonists LILLY CO ELI (US) 2007-05-02 CN disclosed