SCHEMBL4637787

SCHEMBL4637787

ClON=Cc1ccncc1Cl

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.39
HTT P42858 1/20 0.37
CDK5 Q00535 1/20 0.37
CDK5R1 Q15078 1/20 0.37
NFE2L2 Q16236 1/20 0.35
MAPT P10636 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
NFATC1 O95644 1/20 0.30
GSK3B P49841 1/20 0.30
DYRK1A Q13627 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4637909 0.85 GAA (0.35) GAAHTTCDK5CDK5R1MAPT
SCHEMBL4637844 0.77 GAA (0.42) GAAHTTCDK5CDK5R1NFE2L2
SCHEMBL4637840 0.77 GAA (0.42) GAAHTTCDK5CDK5R1NFE2L2
SCHEMBL15741494 0.73
SCHEMBL28618300 0.72 ALDH1A1 (0.50) GAAMAPTNPSR1
SCHEMBL22017330 0.70 HTT (0.41) GAAHTTCDK5CDK5R1NFE2L2
SCHEMBL28657657 0.70 GRIN2D (0.60) MAPTNPSR1
SCHEMBL117895 0.70
SCHEMBL29954572 0.70
SCHEMBL3661431 0.70

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501808-B1 TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-07-02 EP disclosed