SCHEMBL4637852

SCHEMBL4637852

COc1ccc(OC(F)(F)F)cc1Cn1nnc(C(=O)C#Cc2ccccc2Cl)c1-c1cccnc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 4/20 0.40
IDH1 O75874 1/20 0.37
CYP11B1 P15538 2/20 0.35
CYP11B2 P19099 2/20 0.35
SLC16A3 O15427 1/20 0.35
SLC16A1 P53985 1/20 0.35
MCTS1 Q9ULC4 1/20 0.35
CHRM5 P08912 1/20 0.35
CYP19A1 P11511 1/20 0.35
GPR139 Q6DWJ6 1/20 0.34
TACR1 P25103 2/20 0.34
ALDH1A1 P00352 2/20 0.34
KDR P35968 1/20 0.34
F2RL3 Q96RI0 1/20 0.34
LMNA P02545 1/20 0.33
MAPT P10636 1/20 0.33
HPGD P15428 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
HCRTR1 O43613 1/20 0.33
HCRTR2 O43614 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4637847 0.86 ABL1 (0.40) ABL1IDH1CYP11B1CYP11B2SLC16A3
SCHEMBL4637989 0.84 ABL1 (0.47) ABL1CYP11B1CYP11B2CHRM5CYP19A1
SCHEMBL4638893 0.81 ABL1 (0.44) ABL1CYP11B1CYP11B2CHRM5GPR139
SCHEMBL4637714 0.79 IDH1 (0.54) IDH1CYP19A1ALDH1A1
SCHEMBL4707915 0.79 IDH1 (0.48) IDH1CYP19A1ALDH1A1KDR
SCHEMBL6426240 0.79 ABL1 (0.38) ABL1IDH1CYP11B1CYP11B2SLC16A3
SCHEMBL4637753 0.77 IDH1 (0.47) IDH1CYP19A1ALDH1A1MAPTSMN1; SMN2
SCHEMBL4638811 0.77 IDH1 (0.40) IDH1CYP19A1ALDH1A1MAPTSMN1; SMN2
SCHEMBL4638905 0.76 IDH1 (0.41) IDH1CYP19A1ALDH1A1KDRMAPT
SCHEMBL5795131 0.74 ABL1 (0.43) ABL1CYP19A1GPR139TACR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501808-B1 TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-07-02 EP disclosed