SCHEMBL4637847

SCHEMBL4637847

COc1ccc(OC(F)(F)F)cc1Cn1nnc(C#CC(=O)c2ccccc2Cl)c1-c1cccnc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 3/20 0.40
CHRM5 P08912 2/20 0.36
CYP11B1 P15538 3/20 0.36
CYP11B2 P19099 3/20 0.36
ALDH1A1 P00352 2/20 0.35
SLC16A3 O15427 1/20 0.35
SLC16A1 P53985 1/20 0.35
MCTS1 Q9ULC4 1/20 0.35
SGMS2 Q8NHU3 1/20 0.35
TACR1 P25103 2/20 0.34
HTR2C P28335 2/20 0.34
KDR P35968 1/20 0.34
F2RL3 Q96RI0 1/20 0.34
IDH1 O75874 1/20 0.34
CYP1A2 P05177 1/20 0.34
HTR2A P28223 1/20 0.34
HTR2B P41595 1/20 0.34
LMNA P02545 1/20 0.33
MAPT P10636 1/20 0.33
HPGD P15428 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4637852 0.86 ABL1 (0.40) ABL1CHRM5CYP11B1CYP11B2ALDH1A1
SCHEMBL4637989 0.79 ABL1 (0.47) ABL1CHRM5CYP11B1CYP11B2TACR1
SCHEMBL4638481 0.79 IDH1 (0.44) CYP11B1CYP11B2TACR1KDRIDH1
SCHEMBL4637712 0.79 IDH1 (0.51) IDH1MAPTSMN1; SMN2
SCHEMBL4637750 0.77 IDH1 (0.43) IDH1MAPTSMN1; SMN2
SCHEMBL4638808 0.77 P2RX7 (0.38) CYP11B2ALDH1A1IDH1CYP1A2MAPT
SCHEMBL4638903 0.76 IDH1 (0.38) CYP11B1CYP11B2ALDH1A1KDRIDH1
SCHEMBL4638893 0.76 ABL1 (0.44) ABL1CHRM5CYP11B1CYP11B2ALDH1A1
SCHEMBL6426240 0.74 ABL1 (0.38) ABL1CHRM5CYP11B1CYP11B2SLC16A3
SCHEMBL4637948 0.71 RORB (0.36) TACR1IDH1MAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501808-B1 TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-07-02 EP disclosed