SCHEMBL4637872

SCHEMBL4637872

CC(C)(C)[Si](C)(C)OCC#CC(=O)c1nnn(Cc2cc(C(F)(F)F)cc(C(F)(F)F)c2)c1-c1cnccn1

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
USP2 O75604 3/20 0.36
CYP3A4 P08684 2/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
CYP2D6 P10635 2/20 0.35
TSHR P16473 1/20 0.33
P2RX7 Q99572 1/20 0.33
TACR1 P25103 1/20 0.31
AKR1C3 P42330 1/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4639457 0.86 USP2 (0.35) USP2CYP3A4CYP2D6TSHRTACR1
SCHEMBL4637768 0.84 USP2 (0.37) USP2CYP3A4MEN1KMT2ACYP2D6
SCHEMBL4638914 0.83 ALDH1A1 (0.43) TSHRTACR1MAPT
SCHEMBL4708145 0.83 AKR1C3 (0.36) USP2MEN1KMT2ACYP2D6TSHR
SCHEMBL4638494 0.79 USP2 (0.42) USP2CYP3A4MEN1KMT2ACYP2D6
SCHEMBL4637963 0.79 USP2 (0.45) USP2CYP3A4MEN1KMT2ACYP2D6
SCHEMBL4639425 0.78 USP2 (0.35) USP2CYP3A4CYP2D6TSHRTACR1
SCHEMBL4637887 0.76 USP2 (0.36) USP2CYP3A4MEN1KMT2ACYP2D6
SCHEMBL4637960 0.76 USP2 (0.41) USP2CYP3A4MEN1KMT2ACYP2D6
SCHEMBL4638484 0.74 AKR1C3 (0.35) USP2MEN1KMT2ACYP2D6TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501808-B1 TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-07-02 EP disclosed