SCHEMBL4637896

SCHEMBL4637896

Cc1nc(-c2ccccc2Cl)c(Br)o1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.47
MAPT P10636 2/20 0.47
RAB9A P51151 3/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
TP53 P04637 2/20 0.43
HPGD P15428 2/20 0.43
PTGS1 P23219 1/20 0.43
PTGS2 P35354 1/20 0.43
HSD11B1 P28845 2/20 0.41
KMT2A Q03164 5/20 0.40
HSD17B10 Q99714 2/20 0.40
MEN1 O00255 2/20 0.40
POLB P06746 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
KDM4E B2RXH2 2/20 0.39
ALDH1A1 P00352 2/20 0.39
TSHR P16473 1/20 0.39
NFKB1 P19838 1/20 0.39
CASP3 P42574 1/20 0.39
NFKB2 Q00653 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5541542 0.82 MAPT (0.49) NPC1MAPTRAB9ASMN1; SMN2TP53
SCHEMBL5541531 0.79 NPC1 (0.47) NPC1MAPTRAB9ASMN1; SMN2TP53
SCHEMBL4638002 0.79 NPC1 (0.40) NPC1RAB9ASMN1; SMN2TP53HPGD
SCHEMBL10833758 0.79 NPC1 (0.44) NPC1MAPTRAB9ASMN1; SMN2TP53
SCHEMBL4638829 0.74 NPC1 (0.40) NPC1MAPTRAB9ASMN1; SMN2TP53
SCHEMBL31469380 0.74 MAPK13 (0.54) MAPTRAB9ASMN1; SMN2TP53HPGD
SCHEMBL5547946 0.71 NPC1 (0.46) NPC1MAPTRAB9ASMN1; SMN2TP53
SCHEMBL10832282 0.70 KMT2A (0.45) NPC1MAPTKMT2AHSD17B10L3MBTL1
SCHEMBL10832274 0.69 RXRA (0.57) KMT2AHSD17B10
SCHEMBL5547942 0.69 NPC1 (0.43) NPC1MAPTRAB9ASMN1; SMN2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501808-B1 TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-07-02 EP disclosed
CN-1649849-A Tachykinin receptor antagonists LILLY CO ELI (US) 2005-08-03 CN disclosed