SCHEMBL4638829

SCHEMBL4638829

Clc1ccccc1-c1nc(C2CC2)oc1Br

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.40
RAB9A P51151 4/20 0.40
KMT2A Q03164 3/20 0.40
MEN1 O00255 2/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
POLB P06746 1/20 0.40
SMN1; SMN2 Q16637 3/20 0.39
TP53 P04637 2/20 0.39
HPGD P15428 1/20 0.39
GPBAR1 Q8TDU6 2/20 0.38
ALDH1A1 P00352 6/20 0.36
HTT P42858 3/20 0.36
LMNA P02545 2/20 0.36
NPSR1 Q6W5P4 2/20 0.36
MAPT P10636 1/20 0.36
KDM4E B2RXH2 3/20 0.36
TSHR P16473 2/20 0.36
NFKB1 P19838 1/20 0.36
CASP3 P42574 1/20 0.36
NFKB2 Q00653 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4637896 0.74 NPC1 (0.47) NPC1RAB9AKMT2AMEN1L3MBTL1
SCHEMBL4638002 0.71 NPC1 (0.40) NPC1RAB9AKMT2AMEN1L3MBTL1
SCHEMBL4638835 0.69 HSP90AA1 (0.38) NPC1RAB9AL3MBTL1SMN1; SMN2TP53
SCHEMBL24598909 0.67 GPBAR1 (0.48) KMT2AGPBAR1ALDH1A1HTTLMNA
SCHEMBL29692090 0.67 GPBAR1 (0.48) KMT2AGPBAR1ALDH1A1HTTLMNA
SCHEMBL28318365 0.65 HTR3A (0.43) NPC1RAB9AKMT2AMEN1L3MBTL1
SCHEMBL21486108 0.65 USP1 (0.42) NPC1RAB9AKMT2AMEN1POLB
SCHEMBL30605725 0.64 GPBAR1 (0.51) KMT2AGPBAR1ALDH1A1HTTLMNA
SCHEMBL24598908 0.64 GPBAR1 (0.51) KMT2AGPBAR1ALDH1A1HTTLMNA
SCHEMBL21098177 0.64 GPBAR1 (0.54) NPC1KMT2AMEN1GPBAR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501808-B1 TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-07-02 EP disclosed
CN-1649849-A Tachykinin receptor antagonists LILLY CO ELI (US) 2005-08-03 CN disclosed