SCHEMBL4638258

SCHEMBL4638258

CC(C)(C)c1ccc(NC(=O)NNC(=O)O)cc1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 4/20 0.65
EPHX2 P34913 2/20 0.65
RAB9A P51151 4/20 0.62
NPC1 O15118 3/20 0.62
SMN1; SMN2 Q16637 3/20 0.62
MAPT P10636 2/20 0.62
MAPK1 P28482 2/20 0.62
HTT P42858 2/20 0.62
MEN1 O00255 1/20 0.62
XBP1 P17861 1/20 0.62
KMT2A Q03164 1/20 0.62
TRPV1 Q8NER1 3/20 0.58
KIF11 P52732 1/20 0.53
EPHX1 P07099 1/20 0.53
HDAC3 O15379 1/20 0.51
HDAC11 Q96DB2 1/20 0.51
HDAC8 Q9BY41 1/20 0.51
HDAC6 Q9UBN7 1/20 0.51
CNR1 P21554 1/20 0.51
TSHR P16473 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13756246 0.85 MAPT (0.81) NR1H4EPHX2RAB9ANPC1SMN1; SMN2
SCHEMBL2730172 0.85 MAPT (0.81) NR1H4EPHX2RAB9ANPC1SMN1; SMN2
SCHEMBL2090691 0.83 NR1H4 (0.65) NR1H4EPHX2RAB9ANPC1SMN1; SMN2
SCHEMBL12585027 0.81 MAPT (0.71) NR1H4EPHX2RAB9ANPC1SMN1; SMN2
SCHEMBL17072026 0.81 EPHX2 (0.74) NR1H4EPHX2RAB9ANPC1SMN1; SMN2
SCHEMBL10201044 0.79 NPC1 (0.68) NR1H4EPHX2RAB9ANPC1SMN1; SMN2
SCHEMBL22059470 0.79 NR1H4 (1.00) NR1H4EPHX2RAB9ANPC1SMN1; SMN2
SCHEMBL9037064 0.78 NPC1 (0.66) NR1H4EPHX2RAB9ANPC1SMN1; SMN2
SCHEMBL13141239 0.78 NPC1 (0.68) NR1H4EPHX2RAB9ANPC1SMN1; SMN2
SCHEMBL14292513 0.77 RAB9A (0.59) NR1H4EPHX2RAB9ANPC1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1889831-A2 Diazenedicarboxamides as inhibitors of D-alanine: D-alanine ligase (Ddl) University of Ljubljana (SI) 2008-02-20 EP disclosed